2-ARYLINDENES AND 2-ARYLINDENONES - MOLECULAR-STRUCTURES AND CONSIDERATIONS IN THE BINDING ORIENTATION OF UNSYMMETRICAL NONSTEROIDAL LIGANDS TO THE ESTROGEN-RECEPTOR

被引：124

作者：

ANSTEAD, GM ^{[1
]}

WILSON, SR ^{[1
]}

KATZENELLENBOGEN, JA ^{[1
]}

机构：

[1] UNIV ILLINOIS,DEPT CHEM,1209 W CALIF ST,URBANA,IL 61801

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1989年 / 32卷 / 09期

关键词：

D O I：

10.1021/jm00129a024

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：2163 / 2171

页数：9

共 53 条

[1] FUNCTIONAL-GROUP CONTRIBUTIONS TO DRUG RECEPTOR INTERACTIONS [J].

ANDREWS, PR ;

CRAIK, DJ ;

MARTIN, JL .

JOURNAL OF MEDICINAL CHEMISTRY, 1984, 27 (12) :1648-1657

[2] FLUORESCENCE PROPERTIES OF 2,3-DIARYLINDENES [J].

ANSTEAD, GM ;

KATZENELLENBOGEN, JA .

JOURNAL OF PHYSICAL CHEMISTRY, 1988, 92 (22) :6249-6258

[3] OPTIMIZING OF 2,3-DIARYLINDENES AS FLUORESCENT ESTROGENS - VARIATION OF THE ACCEPTOR GROUP, ORTHO SUBSTITUTION OF THE 2-RING, AND C-1 METHYLATION [J].

ANSTEAD, GM ;

KATZENELLENBOGEN, JA .

JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (09) :1754-1761

[4] 2-ARYLINDENES AND 2-ARYLINDENONES - SYNTHESIS OF PROBES TO STUDY THE BINDING ORIENTATION OF UNSYMMETRICAL NONSTEROIDAL LIGANDS TO THE ESTROGEN-RECEPTOR [J].

ANSTEAD, GM ;

ENSIGN, JL ;

PETERSON, CS ;

KATZENELLENBOGEN, JA .

JOURNAL OF ORGANIC CHEMISTRY, 1989, 54 (07) :1485-1491

[5] 2,3-DIARYLINDENES AND 2,3-DIARYLINDENONES - SYNTHESIS, MOLECULAR-STRUCTURE, PHOTOCHEMISTRY, ESTROGEN-RECEPTOR BINDING-AFFINITY, AND COMPARISONS WITH RELATED TRIARYLETHYLENES [J].

ANSTEAD, GM ;

ALTENBACH, RJ ;

WILSON, SR ;

KATZENELLENBOGEN, JA .

JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (07) :1316-1326

[6]

ANSTEAD GM, UNPUB PHOTOCHEM PHOT

[7]

ANSTEAD GM, IN PRESS J STEROID B

[8]

BEDDELL CR, 1984, CHEM SOC REV, V10, P279

[9] REGIO AND STEREOSPECIFIC SYNTHESIS OF 11-BETA-SUBSTITUTED 19-NORSTEROIDS - INFLUENCE OF 11-BETA-SUBSTITUTION ON PROGESTERONE-RECEPTOR AFFINITY [J].

BELANGER, A ;

PHILIBERT, D ;

TEUTSCH, G .

STEROIDS, 1981, 37 (04) :361-382

[10]

BIELLMANN JF, 1986, ACCOUNTS CHEM RES, V19, P121

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