Inhibition and induction of human cytochrome P450 (CYP) enzymes

被引:306
作者
Pelkonen, O [1 ]
Mäenpää, J
Taavitsainen, P
Rautio, A
Raunio, H
机构
[1] Univ Oulu, Dept Pharmacol & Toxicol, FIN-90220 Oulu, Finland
[2] Leiras OY, Clin Res, FIN-00101 Helsinki, Finland
关键词
D O I
10.1080/004982598238886
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:1203 / 1253
页数:51
相关论文
共 267 条
[81]   CYTOCHROME-P450 - ADVANCES AND PROSPECTS [J].
GUENGERICH, FP .
FASEB JOURNAL, 1992, 6 (02) :667-668
[82]   OXIDATION OF TOXIC AND CARCINOGENIC CHEMICALS BY HUMAN CYTOCHROME-P-450 ENZYMES [J].
GUENGERICH, FP ;
SHIMADA, T .
CHEMICAL RESEARCH IN TOXICOLOGY, 1991, 4 (04) :391-407
[83]   MECHANISM-BASED INACTIVATION OF HUMAN LIVER MICROSOMAL CYTOCHROME-P-450-IIIA4 BY GESTODENE [J].
GUENGERICH, FP .
CHEMICAL RESEARCH IN TOXICOLOGY, 1990, 3 (04) :363-371
[84]   Expression of CYP1B1 in human adult and fetal tissues and differential inducibility of CYP1B1 and CYP1A1 by Ah receptor ligands in human placenta and cultured cells [J].
Hakkola, J ;
Pasanen, M ;
Pelkonen, O ;
Hukkanen, J ;
Evisalmi, S ;
Anttila, S ;
Rane, A ;
Mantyla, M ;
Purkunen, R ;
Saarikoski, S ;
Tooming, M ;
Raunio, H .
CARCINOGENESIS, 1997, 18 (02) :391-397
[85]   Regioselective and stereoselective metabolism of ibuprofen by human cytochrome P450 2C [J].
Hamman, MA ;
Thompson, GA ;
Hall, SD .
BIOCHEMICAL PHARMACOLOGY, 1997, 54 (01) :33-41
[86]   THE ARYL-HYDROCARBON RECEPTOR COMPLEX [J].
HANKINSON, O .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1995, 35 :307-340
[87]  
Hardman J.G., 1996, Goodman and Gilman's The Pharmacological Basis of Therapeutics, V9th
[88]  
HARRIS JW, 1994, CANCER RES, V54, P4026
[89]  
Harris M.O., 1995, CHEM ECOLOGY INSECTS, V2, P3
[90]   GENE STRUCTURE OF CYP3A4, AN ADULT-SPECIFIC FORM OF CYTOCHROME-P450 IN HUMAN LIVERS, AND ITS TRANSCRIPTIONAL CONTROL [J].
HASHIMOTO, H ;
TOIDE, K ;
KITAMURA, R ;
FUJITA, M ;
TAGAWA, S ;
ITOH, S ;
KAMATAKI, T .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1993, 218 (02) :585-595