Discovery of a potent, orally active, nonsteroidal androgen receptor agonist: 4-ethyl-1,2,3,4-tetrahydro-6(trifluoromethyl)-8-pyridono[5,6-g]-quinoline (LG121071)

被引：80

作者：

Hamann, LG

Mani, NS

Davis, RL

Wang, XN

Marschke, KB

Jones, TK

机构：

[1] Ligand Pharmaceut Inc, Dept Med Chem, San Diego, CA 92121 USA

[2] Ligand Pharmaceut Inc, Dept Endocrine Res, San Diego, CA 92121 USA

[3] Ligand Pharmaceut Inc, Dept New Leads Discovery, San Diego, CA 92121 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1999年 / 42卷 / 02期

关键词：

D O I：

10.1021/jm9806648

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：210 / 212

页数：3

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