Direct preparation of primary amides from carboxylic acids and urea using imidazole under microwave irradiation

被引：68

作者：

Khalafi-Nezhad, A ^{[1
]}

Mokhtari, B ^{[1
]}

Rad, MNS ^{[1
]}

机构：

[1] Shiraz Univ, Dept Chem, Coll Sci, Shiraz 71454, Iran

来源：

TETRAHEDRON LETTERS | 2003年 / 44卷 / 39期

关键词：

D O I：

10.1016/S0040-4039(03)01866-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 [有机化学]; 081704 [应用化学];

摘要：

A very simple and efficient solvent-free procedure for the preparation of primary amides is described from carboxylic acids and urea using imidazole under microwave irradiation. Various aliphatic and aromatic primary amides were prepared in good yields by this direct amidation method. (C) 2003 Elsevier Ltd. All rights reserved.

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收藏

页码：7325 / 7328

页数：4

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