Sodium channel modifiers from scorpion venom: Structure-activity relationship, mode of action and application

被引:30
作者
Gurevitz, M [1 ]
Froy, O
Zilberberg, N
Turkov, M
Strugatsky, D
Gershburg, E
Lee, D
Adams, ME
机构
[1] Tel Aviv Univ, Fac Life Sci, Dept Plant Sci, IL-69978 Tel Aviv, Israel
[2] Univ Calif Riverside, Dept Entomol, Riverside, CA 92521 USA
[3] Weizmann Inst Sci, Dept Biol Struct, IL-76100 Rehovot, Israel
[4] Hebrew Univ Jerusalem, Inst Life Sci, Dept Biol Chem, IL-91904 Jerusalem, Israel
[5] CNRS, UPR 9027, IBSM, F-13402 Marseille 20, France
[6] Nicholas Copernicus Univ, Inst Biol & Protect Environm, Biophys Lab, Torun, Poland
[7] Univ Angers, Fac Med, Neurophysiol Lab, F-49045 Angers, France
[8] CEA Saclay, Dept Ingn & Etud Prot, F-91191 Gif Sur Yvette, France
[9] Agr Res Org, Volcani Ctr, Inst Plant Protect, IL-50250 Bet Dagan, Israel
关键词
D O I
10.1016/S0041-0101(98)00160-3
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:1671 / 1682
页数:12
相关论文
共 62 条
[31]   PRIMARY STRUCTURE OF SCORPION ANTIINSECT TOXINS ISOLATED FROM THE VENOM OF LEIURUS-QUINQUESTRIATUS-QUINQUESTRIATUS [J].
KOPEYAN, C ;
MANSUELLE, P ;
SAMPIERI, F ;
BRANDO, T ;
BAHRAOUI, EM ;
ROCHAT, H ;
GRANIER, C .
FEBS LETTERS, 1990, 261 (02) :423-426
[32]   EFFECT OF SCORPION VENOM ON IONIC CURRENTS OF NODE RANVIER .I. PERMEABILITIES PNA AND PK [J].
KOPPENHOFER, E ;
SCHMIDT, H .
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 1968, 303 (02) :133-+
[33]   EFFECT OF SCORPION VENOM ON IONIC CURRENTS OF NODE OF RANVIER .2. INCOMPLETE SODIUM INACTIVATION [J].
KOPPENHOFER, E ;
SCHMIDT, H .
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 1968, 303 (02) :150-+
[34]   H-1-NMR-derived secondary structure and the overall fold of the potent anti-mammal and anti-insect toxin III from the scorpion Leiurus quinquestriatus quinquestriatus [J].
Landon, C ;
Cornet, B ;
Bonmatin, JM ;
Kopeyan, C ;
Rochat, H ;
Vovelle, F ;
Ptak, M .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1996, 236 (02) :395-404
[35]  
LEE D, UNPUB SYNAPTIC ACTIO
[36]   PURIFICATION, CHARACTERIZATION AND ACTION OF 2 INSECT TOXINS FROM THE VENOM OF THE SCORPION BUTHOTUS-JUDAICUS [J].
LESTER, D ;
LAZAROVICI, P ;
PELHATE, M ;
ZLOTKIN, E .
BIOCHIMICA ET BIOPHYSICA ACTA, 1982, 701 (03) :370-381
[37]   INTERACTION OF INSECTICIDES OF THE PYRETHROID FAMILY WITH SPECIFIC BINDING-SITES ON THE VOLTAGE-DEPENDENT SODIUM-CHANNEL FROM MAMMALIAN BRAIN [J].
LOMBET, A ;
MOURRE, C ;
LAZDUNSKI, M .
BRAIN RESEARCH, 1988, 459 (01) :44-53
[38]   INSECTICIDAL EFFECTS OF AN INSECT-SPECIFIC NEUROTOXIN EXPRESSED BY A RECOMBINANT BACULOVIRUS [J].
MAEDA, S ;
VOLRATH, SL ;
HANZLIK, TN ;
HARPER, SA ;
KEI, MM ;
MADDOX, DW ;
HAMMOCK, BD ;
FOWLER, E .
VIROLOGY, 1991, 184 (02) :777-780
[39]  
Martin-Eauclaire M. F., 1995, Handbook of neurotoxicology., P683
[40]  
MCCUTCHEN BF, 1991, BIO-TECHNOL, V9, P848, DOI 10.1038/nbt0991-848