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In vitro assessment of human cytochrome P450
被引:108
作者
:
Clarke, SE
论文数:
0
引用数:
0
h-index:
0
机构:
SmithKline Beecham Pharmaceut, Drug Metab & Pharmacokinet, Welwyn Garden City AL6 9AR, Herts, England
SmithKline Beecham Pharmaceut, Drug Metab & Pharmacokinet, Welwyn Garden City AL6 9AR, Herts, England
Clarke, SE
[
1
]
机构
:
[1]
SmithKline Beecham Pharmaceut, Drug Metab & Pharmacokinet, Welwyn Garden City AL6 9AR, Herts, England
来源
:
XENOBIOTICA
|
1998年
/ 28卷
/ 12期
关键词
:
D O I
:
10.1080/004982598238877
中图分类号
:
R9 [药学];
学科分类号
:
1007 ;
摘要
:
[No abstract available]
引用
收藏
页码:1167 / 1202
页数:36
相关论文
共 213 条
[151]
RODRIGUES AD, 1995, DRUG METAB DISPOS, V23, P765
[152]
CLONING AND EXPRESSION OF COMPLEMENTARY DNAS FOR MULTIPLE MEMBERS OF THE HUMAN CYTOCHROME-P450IIC SUBFAMILY
ROMKES, M
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,RES TRIANGLE PK,NC 27709
ROMKES, M
FALETTO, MB
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,RES TRIANGLE PK,NC 27709
FALETTO, MB
BLAISDELL, JA
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,RES TRIANGLE PK,NC 27709
BLAISDELL, JA
RAUCY, JL
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,RES TRIANGLE PK,NC 27709
RAUCY, JL
GOLDSTEIN, JA
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,RES TRIANGLE PK,NC 27709
GOLDSTEIN, JA
[J].
BIOCHEMISTRY,
1991,
30
(13)
: 3247
-
3255
[153]
PURIFICATION AND CHARACTERIZATION OF HEPATIC-MICROSOMAL CYTOCHROME-P-450
RYAN, DE
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Protein Biochemistry, Hoffmann-La Roche Inc., Nutley
RYAN, DE
LEVIN, W
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Protein Biochemistry, Hoffmann-La Roche Inc., Nutley
LEVIN, W
[J].
PHARMACOLOGY & THERAPEUTICS,
1990,
45
(02)
: 153
-
239
[154]
EXPRESSION OF MODIFIED HUMAN CYTOCHROME-P450 1A2 IN ESCHERICHIA-COLI - STABILIZATION, PURIFICATION, SPECTRAL CHARACTERIZATION, AND CATALYTIC ACTIVITIES OF THE ENZYME
SANDHU, P
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
SANDHU, P
GUO, ZY
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
GUO, ZY
BABA, T
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
BABA, T
MARTIN, MV
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
MARTIN, MV
TUKEY, RH
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
TUKEY, RH
GUENGERICH, FP
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
GUENGERICH, FP
[J].
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS,
1994,
309
(01)
: 168
-
177
[155]
EXPRESSION OF MODIFIED CYTOCHROME-P450-2C10-(2C9) IN ESCHERICHIA-COLI, PURIFICATION, AND RECONSTITUTION OF CATALYTIC ACTIVITY
SANDHU, P
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,MED CTR,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
SANDHU, P
BABA, T
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,MED CTR,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
BABA, T
GUENGERICH, FP
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,MED CTR,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
GUENGERICH, FP
[J].
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS,
1993,
306
(02)
: 443
-
450
[156]
INVITRO EFFECT OF FLUOROQUINOLONES ON THEOPHYLLINE METABOLISM IN HUMAN LIVER-MICROSOMES
SARKAR, M
论文数:
0
引用数:
0
h-index:
0
机构:
VIRGINIA COMMONWEALTH UNIV, MED COLL VIRGINIA, SCH PHARM, DEPT PHARM & PHARMACEUT, RICHMOND, VA 23298 USA
SARKAR, M
POLK, RE
论文数:
0
引用数:
0
h-index:
0
机构:
VIRGINIA COMMONWEALTH UNIV, MED COLL VIRGINIA, SCH PHARM, DEPT PHARM & PHARMACEUT, RICHMOND, VA 23298 USA
POLK, RE
GUZELIAN, PS
论文数:
0
引用数:
0
h-index:
0
机构:
VIRGINIA COMMONWEALTH UNIV, MED COLL VIRGINIA, SCH PHARM, DEPT PHARM & PHARMACEUT, RICHMOND, VA 23298 USA
GUZELIAN, PS
HUNT, C
论文数:
0
引用数:
0
h-index:
0
机构:
VIRGINIA COMMONWEALTH UNIV, MED COLL VIRGINIA, SCH PHARM, DEPT PHARM & PHARMACEUT, RICHMOND, VA 23298 USA
HUNT, C
KARNES, HT
论文数:
0
引用数:
0
h-index:
0
机构:
VIRGINIA COMMONWEALTH UNIV, MED COLL VIRGINIA, SCH PHARM, DEPT PHARM & PHARMACEUT, RICHMOND, VA 23298 USA
KARNES, HT
[J].
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY,
1990,
34
(04)
: 594
-
599
[157]
EXPRESSION OF CYP1A1 AND CYP1A2 GENES IN HUMAN LIVER
SCHWEIKL, H
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,POB 12233,RES TRIANGLE PK,NC 27709
SCHWEIKL, H
TAYLOR, JA
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,POB 12233,RES TRIANGLE PK,NC 27709
TAYLOR, JA
KITAREEWAN, S
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,POB 12233,RES TRIANGLE PK,NC 27709
KITAREEWAN, S
LINKO, P
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,POB 12233,RES TRIANGLE PK,NC 27709
LINKO, P
NAGORNEY, D
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,POB 12233,RES TRIANGLE PK,NC 27709
NAGORNEY, D
GOLDSTEIN, JA
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,POB 12233,RES TRIANGLE PK,NC 27709
GOLDSTEIN, JA
[J].
PHARMACOGENETICS,
1993,
3
(05):
: 239
-
249
[158]
HIGH PROMUTAGEN ACTIVATING CAPACITY OF YEAST MICROSOMES CONTAINING HUMAN CYTOCHROME-P-450 1A AND HUMAN NADPH-CYTOCHROME P-450 REDUCTASE
SENGSTAG, C
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ZURICH, CH-8603 SCHWERZENBACH, SWITZERLAND
UNIV ZURICH, CH-8603 SCHWERZENBACH, SWITZERLAND
SENGSTAG, C
EUGSTER, HP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ZURICH, CH-8603 SCHWERZENBACH, SWITZERLAND
UNIV ZURICH, CH-8603 SCHWERZENBACH, SWITZERLAND
EUGSTER, HP
WURGLER, FE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ZURICH, CH-8603 SCHWERZENBACH, SWITZERLAND
UNIV ZURICH, CH-8603 SCHWERZENBACH, SWITZERLAND
WURGLER, FE
[J].
CARCINOGENESIS,
1994,
15
(05)
: 837
-
843
[159]
A FORM OF CYTOCHROME-P450 IN MAN, ORTHOLOGOUS TO FORM D IN THE RAT, CATALYZES THE O-DEETHYLATION OF PHENACETIN AND IS INDUCIBLE BY CIGARETTE-SMOKING
SESARDIC, D
论文数:
0
引用数:
0
h-index:
0
SESARDIC, D
BOOBIS, AR
论文数:
0
引用数:
0
h-index:
0
BOOBIS, AR
EDWARDS, RJ
论文数:
0
引用数:
0
h-index:
0
EDWARDS, RJ
DAVIES, DS
论文数:
0
引用数:
0
h-index:
0
DAVIES, DS
[J].
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY,
1988,
26
(04)
: 363
-
372
[160]
FURAFYLLINE IS A POTENT AND SELECTIVE INHIBITOR OF CYTOCHROME-P450IA2 IN MAN
SESARDIC, D
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL POSTGRAD MED SCH,DEPT CLIN PHARMACOL,LONDON W12 0NN,ENGLAND
SESARDIC, D
BOOBIS, AR
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL POSTGRAD MED SCH,DEPT CLIN PHARMACOL,LONDON W12 0NN,ENGLAND
BOOBIS, AR
MURRAY, BP
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL POSTGRAD MED SCH,DEPT CLIN PHARMACOL,LONDON W12 0NN,ENGLAND
MURRAY, BP
MURRAY, S
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL POSTGRAD MED SCH,DEPT CLIN PHARMACOL,LONDON W12 0NN,ENGLAND
MURRAY, S
SEGURA, J
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL POSTGRAD MED SCH,DEPT CLIN PHARMACOL,LONDON W12 0NN,ENGLAND
SEGURA, J
DELATORRE, R
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL POSTGRAD MED SCH,DEPT CLIN PHARMACOL,LONDON W12 0NN,ENGLAND
DELATORRE, R
DAVIES, DS
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL POSTGRAD MED SCH,DEPT CLIN PHARMACOL,LONDON W12 0NN,ENGLAND
DAVIES, DS
[J].
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY,
1990,
29
(06)
: 651
-
663
←
11
12
13
14
15
16
17
18
19
20
→
共 213 条
[151]
RODRIGUES AD, 1995, DRUG METAB DISPOS, V23, P765
[152]
CLONING AND EXPRESSION OF COMPLEMENTARY DNAS FOR MULTIPLE MEMBERS OF THE HUMAN CYTOCHROME-P450IIC SUBFAMILY
ROMKES, M
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,RES TRIANGLE PK,NC 27709
ROMKES, M
FALETTO, MB
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,RES TRIANGLE PK,NC 27709
FALETTO, MB
BLAISDELL, JA
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,RES TRIANGLE PK,NC 27709
BLAISDELL, JA
RAUCY, JL
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,RES TRIANGLE PK,NC 27709
RAUCY, JL
GOLDSTEIN, JA
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,RES TRIANGLE PK,NC 27709
GOLDSTEIN, JA
[J].
BIOCHEMISTRY,
1991,
30
(13)
: 3247
-
3255
[153]
PURIFICATION AND CHARACTERIZATION OF HEPATIC-MICROSOMAL CYTOCHROME-P-450
RYAN, DE
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Protein Biochemistry, Hoffmann-La Roche Inc., Nutley
RYAN, DE
LEVIN, W
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Protein Biochemistry, Hoffmann-La Roche Inc., Nutley
LEVIN, W
[J].
PHARMACOLOGY & THERAPEUTICS,
1990,
45
(02)
: 153
-
239
[154]
EXPRESSION OF MODIFIED HUMAN CYTOCHROME-P450 1A2 IN ESCHERICHIA-COLI - STABILIZATION, PURIFICATION, SPECTRAL CHARACTERIZATION, AND CATALYTIC ACTIVITIES OF THE ENZYME
SANDHU, P
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
SANDHU, P
GUO, ZY
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
GUO, ZY
BABA, T
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
BABA, T
MARTIN, MV
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
MARTIN, MV
TUKEY, RH
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
TUKEY, RH
GUENGERICH, FP
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
GUENGERICH, FP
[J].
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS,
1994,
309
(01)
: 168
-
177
[155]
EXPRESSION OF MODIFIED CYTOCHROME-P450-2C10-(2C9) IN ESCHERICHIA-COLI, PURIFICATION, AND RECONSTITUTION OF CATALYTIC ACTIVITY
SANDHU, P
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,MED CTR,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
SANDHU, P
BABA, T
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,MED CTR,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
BABA, T
GUENGERICH, FP
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,MED CTR,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
GUENGERICH, FP
[J].
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS,
1993,
306
(02)
: 443
-
450
[156]
INVITRO EFFECT OF FLUOROQUINOLONES ON THEOPHYLLINE METABOLISM IN HUMAN LIVER-MICROSOMES
SARKAR, M
论文数:
0
引用数:
0
h-index:
0
机构:
VIRGINIA COMMONWEALTH UNIV, MED COLL VIRGINIA, SCH PHARM, DEPT PHARM & PHARMACEUT, RICHMOND, VA 23298 USA
SARKAR, M
POLK, RE
论文数:
0
引用数:
0
h-index:
0
机构:
VIRGINIA COMMONWEALTH UNIV, MED COLL VIRGINIA, SCH PHARM, DEPT PHARM & PHARMACEUT, RICHMOND, VA 23298 USA
POLK, RE
GUZELIAN, PS
论文数:
0
引用数:
0
h-index:
0
机构:
VIRGINIA COMMONWEALTH UNIV, MED COLL VIRGINIA, SCH PHARM, DEPT PHARM & PHARMACEUT, RICHMOND, VA 23298 USA
GUZELIAN, PS
HUNT, C
论文数:
0
引用数:
0
h-index:
0
机构:
VIRGINIA COMMONWEALTH UNIV, MED COLL VIRGINIA, SCH PHARM, DEPT PHARM & PHARMACEUT, RICHMOND, VA 23298 USA
HUNT, C
KARNES, HT
论文数:
0
引用数:
0
h-index:
0
机构:
VIRGINIA COMMONWEALTH UNIV, MED COLL VIRGINIA, SCH PHARM, DEPT PHARM & PHARMACEUT, RICHMOND, VA 23298 USA
KARNES, HT
[J].
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY,
1990,
34
(04)
: 594
-
599
[157]
EXPRESSION OF CYP1A1 AND CYP1A2 GENES IN HUMAN LIVER
SCHWEIKL, H
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,POB 12233,RES TRIANGLE PK,NC 27709
SCHWEIKL, H
TAYLOR, JA
论文数:
0
引用数:
0
h-index:
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机构:
NIEHS,BIOCHEM RISK ANAL LAB,POB 12233,RES TRIANGLE PK,NC 27709
TAYLOR, JA
KITAREEWAN, S
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引用数:
0
h-index:
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机构:
NIEHS,BIOCHEM RISK ANAL LAB,POB 12233,RES TRIANGLE PK,NC 27709
KITAREEWAN, S
LINKO, P
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,POB 12233,RES TRIANGLE PK,NC 27709
LINKO, P
NAGORNEY, D
论文数:
0
引用数:
0
h-index:
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机构:
NIEHS,BIOCHEM RISK ANAL LAB,POB 12233,RES TRIANGLE PK,NC 27709
NAGORNEY, D
GOLDSTEIN, JA
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS,BIOCHEM RISK ANAL LAB,POB 12233,RES TRIANGLE PK,NC 27709
GOLDSTEIN, JA
[J].
PHARMACOGENETICS,
1993,
3
(05):
: 239
-
249
[158]
HIGH PROMUTAGEN ACTIVATING CAPACITY OF YEAST MICROSOMES CONTAINING HUMAN CYTOCHROME-P-450 1A AND HUMAN NADPH-CYTOCHROME P-450 REDUCTASE
SENGSTAG, C
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ZURICH, CH-8603 SCHWERZENBACH, SWITZERLAND
UNIV ZURICH, CH-8603 SCHWERZENBACH, SWITZERLAND
SENGSTAG, C
EUGSTER, HP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ZURICH, CH-8603 SCHWERZENBACH, SWITZERLAND
UNIV ZURICH, CH-8603 SCHWERZENBACH, SWITZERLAND
EUGSTER, HP
WURGLER, FE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ZURICH, CH-8603 SCHWERZENBACH, SWITZERLAND
UNIV ZURICH, CH-8603 SCHWERZENBACH, SWITZERLAND
WURGLER, FE
[J].
CARCINOGENESIS,
1994,
15
(05)
: 837
-
843
[159]
A FORM OF CYTOCHROME-P450 IN MAN, ORTHOLOGOUS TO FORM D IN THE RAT, CATALYZES THE O-DEETHYLATION OF PHENACETIN AND IS INDUCIBLE BY CIGARETTE-SMOKING
SESARDIC, D
论文数:
0
引用数:
0
h-index:
0
SESARDIC, D
BOOBIS, AR
论文数:
0
引用数:
0
h-index:
0
BOOBIS, AR
EDWARDS, RJ
论文数:
0
引用数:
0
h-index:
0
EDWARDS, RJ
DAVIES, DS
论文数:
0
引用数:
0
h-index:
0
DAVIES, DS
[J].
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY,
1988,
26
(04)
: 363
-
372
[160]
FURAFYLLINE IS A POTENT AND SELECTIVE INHIBITOR OF CYTOCHROME-P450IA2 IN MAN
SESARDIC, D
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL POSTGRAD MED SCH,DEPT CLIN PHARMACOL,LONDON W12 0NN,ENGLAND
SESARDIC, D
BOOBIS, AR
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL POSTGRAD MED SCH,DEPT CLIN PHARMACOL,LONDON W12 0NN,ENGLAND
BOOBIS, AR
MURRAY, BP
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL POSTGRAD MED SCH,DEPT CLIN PHARMACOL,LONDON W12 0NN,ENGLAND
MURRAY, BP
MURRAY, S
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL POSTGRAD MED SCH,DEPT CLIN PHARMACOL,LONDON W12 0NN,ENGLAND
MURRAY, S
SEGURA, J
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL POSTGRAD MED SCH,DEPT CLIN PHARMACOL,LONDON W12 0NN,ENGLAND
SEGURA, J
DELATORRE, R
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL POSTGRAD MED SCH,DEPT CLIN PHARMACOL,LONDON W12 0NN,ENGLAND
DELATORRE, R
DAVIES, DS
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL POSTGRAD MED SCH,DEPT CLIN PHARMACOL,LONDON W12 0NN,ENGLAND
DAVIES, DS
[J].
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY,
1990,
29
(06)
: 651
-
663
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