Resistance to human immunodeficiency virus type 1 protease inhibitors

被引:160
作者
Boden, D [1 ]
Markowitz, M [1 ]
机构
[1] Aaron Diamond AIDS Res Ctr, New York, NY 10016 USA
关键词
D O I
10.1128/AAC.42.11.2775
中图分类号
Q93 [微生物学];
学科分类号
071005 ; 100705 ;
摘要
引用
收藏
页码:2775 / 2783
页数:9
相关论文
共 97 条
[1]  
[Anonymous], ESPRIT CACID
[2]   DESIGN OF ENZYME-INHIBITORS USING ITERATIVE PROTEIN CRYSTALLOGRAPHIC ANALYSIS [J].
APPELT, K ;
BACQUET, RJ ;
BARTLETT, CA ;
BOOTH, CLJ ;
FREER, ST ;
FUHRY, MAM ;
GEHRING, MR ;
HERRMANN, SM ;
HOWLAND, EF ;
JANSON, CA ;
JONES, TR ;
KAN, CC ;
KATHARDEKAR, V ;
LEWIS, KK ;
MARZONI, GP ;
MATTHEWS, DA ;
MOHR, C ;
MOOMAW, EW ;
MORSE, CA ;
OATLEY, SJ ;
OGDEN, RC ;
REDDY, MR ;
REICH, SH ;
SCHOETTLIN, WS ;
SMITH, WW ;
VARNEY, MD ;
VILLAFRANCA, JE ;
WARD, RW ;
WEBBER, S ;
WEBBER, SE ;
WELSH, KM ;
WHITE, J .
JOURNAL OF MEDICINAL CHEMISTRY, 1991, 34 (07) :1925-1934
[3]  
CAMERON DW, UNPUB RITONAVIR SAQU
[4]   THE HUMAN LUMICAN GENE - ORGANIZATION, CHROMOSOMAL, LOCATION, AND EXPRESSION IN ARTICULAR-CARTILAGE [J].
GROVER, J ;
CHEN, XN ;
KORENBERG, JR ;
ROUGHLEY, PJ .
JOURNAL OF BIOLOGICAL CHEMISTRY, 1995, 270 (37) :21942-21949
[6]   HIV POPULATION-DYNAMICS IN-VIVO - IMPLICATIONS FOR GENETIC-VARIATION, PATHOGENESIS, AND THERAPY [J].
COFFIN, JM .
SCIENCE, 1995, 267 (5197) :483-489
[7]   Treatment of human immunodeficiency virus infection with saquinavir, zidovudine, and zalcitabine [J].
Collier, AC ;
Coombs, RW ;
Schoenfeld, DA ;
Bassett, RL ;
Timpone, J ;
Baruch, A ;
Jones, M ;
Facey, K ;
Whitacre, C ;
McAuliffe, VJ ;
Friedman, HM ;
Merigan, TC ;
Reichman, RC ;
Hooper, C ;
Corey, L .
NEW ENGLAND JOURNAL OF MEDICINE, 1996, 334 (16) :1011-1017
[8]   FLAP OPENING IN HIV-1 PROTEASE SIMULATED BY ACTIVATED MOLECULAR-DYNAMICS [J].
COLLINS, JR ;
BURT, SK ;
ERICKSON, JW .
NATURE STRUCTURAL BIOLOGY, 1995, 2 (04) :334-338
[9]  
COLLINS JR, 1995, ADV EXP MED BIOL, V362, P455
[10]   Genetic correlates of in vivo viral resistance to indinavir, a human immunodeficiency virus type 1 protease inhibitor [J].
Condra, JH ;
Holder, DJ ;
Schleif, WA ;
Blahy, OM ;
Danovich, RM ;
Gabryelski, LJ ;
Graham, DJ ;
Laird, D ;
Quintero, JC ;
Rhodes, A ;
Robbins, HL ;
Roth, E ;
Shivaprakash, M ;
Yang, T ;
Chodakewitz, JA ;
Deutsch, PJ ;
Leavitt, RY ;
Massari, FE ;
Mellors, JW ;
Squires, KE ;
Steigbigel, RT ;
Teppler, H ;
Emini, EA .
JOURNAL OF VIROLOGY, 1996, 70 (12) :8270-8276