Discovery of a novel series of selective MMP inhibitors:: Identification of the γ-sulfone-thiols

被引：33

作者：

Freskos, JN

Mischke, BV

DeCrescenzo, GA

Heintz, R

Getman, DP

Howard, SC

Kishore, NN

McDonald, JJ

Munie, GE

Rangwala, S

Swearingen, CA

Voliva, C

Welsch, DJ

机构：

[1] Searle Discovery Res, Dept Med Oncol, St Louis, MO 63198 USA

[2] Searle Discovery Res, Dept Inflammat Oncol, St Louis, MO 63198 USA

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1999年 / 9卷 / 07期

关键词：

enzyme inhibitors; antitumour compounds;

D O I：

10.1016/S0960-894X(99)00116-X

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：943 / 948

页数：6

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