Efficient Copper-Catalyzed Synthesis of Fused Pyridoquinazolones

被引：7

作者：

Chen, Lujun ^{[1
,2
]}

Fu, Hua ^{[1
]}

Qiao, Renzhong ^{[2
]}

机构：

[1] Tsinghua Univ, Dept Chem, Minist Educ, Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R China

[2] Beijing Univ Chem Technol, Coll Life Sci & Technol, Dept Pharmaceut Engn, State Key Lab Chem Resource Engn, Beijing 100029, Peoples R China

来源：

SYNLETT | 2011年 / 13期

基金：

中国国家自然科学基金;

关键词：

N-heterocycle; pyridoquinazolone; copper; synthetic method; NITROGEN-CONTAINING HETEROCYCLES; COUPLING REACTIONS; N-ARYLATION; C-O; ARYL HALIDES; PRIVILEGED STRUCTURES; CASCADE SYNTHESIS; ROOM-TEMPERATURE; DERIVATIVES; ULLMANN;

D O I：

10.1055/s-0030-1260968

中图分类号：

O62 [有机化学];

学科分类号：

070303 [有机化学];

摘要：

A simple and efficient copper-catalyzed method for synthesis of fused pyridoquinazolones has been developed without addition of any ligand or additive, and it can tolerate various functional groups.

引用

收藏

页码：1930 / 1936

页数：7

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