Histamine H3 Receptor as a Drug Discovery Target

被引:139
作者
Berlin, Michael [1 ]
Boyce, Christopher W. [1 ]
Ruiz, Manuel de Lera [1 ]
机构
[1] Merck Res Labs, Chem Res, Kenilworth, NJ 07033 USA
关键词
ATTENTION-DEFICIT/HYPERACTIVITY DISORDER; CORTICAL ACETYLCHOLINE-RELEASE; PIG PERFUSED BRONCHIOLES; IN-VIVO; PHARMACOLOGICAL CHARACTERIZATION; SUBSTANCE-P; H-3-RECEPTOR ANTAGONIST; COGNITIVE PERFORMANCE; MEDICINAL CHEMISTRY; H3; RECEPTOR;
D O I
10.1021/jm100064d
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:26 / 53
页数:28
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