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Protean agonists - Keys to receptor active states?
被引:24
作者
:
Kenakin, T
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Receptor Biochemistry, GlaxoWellcome, Research Triangle Park, NC 27709
Kenakin, T
机构
:
[1]
Department of Receptor Biochemistry, GlaxoWellcome, Research Triangle Park, NC 27709
来源
:
RECEPTOR CLASSIFICATION: THE INTEGRATION OF OPERATIONAL, STRUCTURAL, AND TRANSDUCTIONAL INFORMATION
|
1997年
/ 812卷
关键词
:
D O I
:
10.1111/j.1749-6632.1997.tb48151.x
中图分类号
:
Q5 [生物化学];
Q7 [分子生物学];
学科分类号
:
071010 ;
081704 ;
摘要
:
[No abstract available]
引用
收藏
页码:116 / 125
页数:10
相关论文
共 16 条
[1]
CHIDIAC P, 1994, MOL PHARMACOL, V45, P490
[2]
ANTAGONISTS WITH NEGATIVE INTRINSIC ACTIVITY AT DELTA-OPIOID RECEPTORS COUPLED TO GTP-BINDING PROTEINS
COSTA, T
论文数:
0
引用数:
0
h-index:
0
机构:
MAX PLANCK INST PSYCHIAT, DEPT NEUROPHARMACOL, D-8033 MARTINSRIED, GERMANY
MAX PLANCK INST PSYCHIAT, DEPT NEUROPHARMACOL, D-8033 MARTINSRIED, GERMANY
COSTA, T
HERZ, A
论文数:
0
引用数:
0
h-index:
0
机构:
MAX PLANCK INST PSYCHIAT, DEPT NEUROPHARMACOL, D-8033 MARTINSRIED, GERMANY
MAX PLANCK INST PSYCHIAT, DEPT NEUROPHARMACOL, D-8033 MARTINSRIED, GERMANY
HERZ, A
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1989,
86
(19)
: 7321
-
7325
[3]
COSTA T, 1992, MOL PHARMACOL, V41, P549
[4]
THE ENERGY LANDSCAPES AND MOTIONS OF PROTEINS
FRAUENFELDER, H
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ILLINOIS, BECKMAN INST, URBANA, IL 61801 USA
UNIV ILLINOIS, BECKMAN INST, URBANA, IL 61801 USA
FRAUENFELDER, H
SLIGAR, SG
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ILLINOIS, BECKMAN INST, URBANA, IL 61801 USA
UNIV ILLINOIS, BECKMAN INST, URBANA, IL 61801 USA
SLIGAR, SG
WOLYNES, PG
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ILLINOIS, BECKMAN INST, URBANA, IL 61801 USA
UNIV ILLINOIS, BECKMAN INST, URBANA, IL 61801 USA
WOLYNES, PG
[J].
SCIENCE,
1991,
254
(5038)
: 1598
-
1603
[5]
FRAUENFELDER H, 1988, ANNU REV BIOPHYS BIO, V17, P451
[6]
SELECTIVE ACTIVATION OF INHIBITORY G-PROTEIN ALPHA-SUBUNITS BY PARTIAL AGONISTS OF THE HUMAN 5-HT(1A) RECEPTOR
GETTYS, TW
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV, MED CTR, DEPT MED, DURHAM, NC 27710 USA
GETTYS, TW
FIELDS, TA
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV, MED CTR, DEPT MED, DURHAM, NC 27710 USA
FIELDS, TA
RAYMOND, JR
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV, MED CTR, DEPT MED, DURHAM, NC 27710 USA
RAYMOND, JR
[J].
BIOCHEMISTRY,
1994,
33
(14)
: 4283
-
4290
[7]
AGONIST-RECEPTOR EFFICACY .2. AGONIST TRAFFICKING OF RECEPTOR SIGNALS
KENAKIN, T
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Cellular Biochemistry, Glaxo Research Institute, Research Triangle Park, NC 27709, Five Moore Drive
KENAKIN, T
[J].
TRENDS IN PHARMACOLOGICAL SCIENCES,
1995,
16
(07)
: 232
-
238
[8]
AGONIST-RECEPTOR EFFICACY .1. MECHANISMS OF EFFICACY AND RECEPTOR PROMISCUITY
KENAKIN, T
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Cellular Biochemistry, Glaxo Research Institute, Research Triangle Park, NC 27709, Five Moore Drive
KENAKIN, T
[J].
TRENDS IN PHARMACOLOGICAL SCIENCES,
1995,
16
(06)
: 188
-
192
[9]
AGONIST-SPECIFIC COUPLING OF A CLONED DROSOPHILA OCTOPAMINE TYRAMINE RECEPTOR TO MULTIPLE 2ND MESSENGER SYSTEMS
ROBB, S
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,DEPT ZOOL,AFRC,MOLEC SIGNALLING LAB,CAMBRIDGE CB2 3EJ,ENGLAND
ROBB, S
CHEEK, TR
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,DEPT ZOOL,AFRC,MOLEC SIGNALLING LAB,CAMBRIDGE CB2 3EJ,ENGLAND
CHEEK, TR
HANNAN, FL
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,DEPT ZOOL,AFRC,MOLEC SIGNALLING LAB,CAMBRIDGE CB2 3EJ,ENGLAND
HANNAN, FL
HALL, LM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,DEPT ZOOL,AFRC,MOLEC SIGNALLING LAB,CAMBRIDGE CB2 3EJ,ENGLAND
HALL, LM
MIDGLEY, JM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,DEPT ZOOL,AFRC,MOLEC SIGNALLING LAB,CAMBRIDGE CB2 3EJ,ENGLAND
MIDGLEY, JM
EVANS, PD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,DEPT ZOOL,AFRC,MOLEC SIGNALLING LAB,CAMBRIDGE CB2 3EJ,ENGLAND
EVANS, PD
[J].
EMBO JOURNAL,
1994,
13
(06)
: 1325
-
1330
[10]
SAMAMA P, 1993, J BIOL CHEM, V268, P4625
←
1
2
→
共 16 条
[1]
CHIDIAC P, 1994, MOL PHARMACOL, V45, P490
[2]
ANTAGONISTS WITH NEGATIVE INTRINSIC ACTIVITY AT DELTA-OPIOID RECEPTORS COUPLED TO GTP-BINDING PROTEINS
COSTA, T
论文数:
0
引用数:
0
h-index:
0
机构:
MAX PLANCK INST PSYCHIAT, DEPT NEUROPHARMACOL, D-8033 MARTINSRIED, GERMANY
MAX PLANCK INST PSYCHIAT, DEPT NEUROPHARMACOL, D-8033 MARTINSRIED, GERMANY
COSTA, T
HERZ, A
论文数:
0
引用数:
0
h-index:
0
机构:
MAX PLANCK INST PSYCHIAT, DEPT NEUROPHARMACOL, D-8033 MARTINSRIED, GERMANY
MAX PLANCK INST PSYCHIAT, DEPT NEUROPHARMACOL, D-8033 MARTINSRIED, GERMANY
HERZ, A
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1989,
86
(19)
: 7321
-
7325
[3]
COSTA T, 1992, MOL PHARMACOL, V41, P549
[4]
THE ENERGY LANDSCAPES AND MOTIONS OF PROTEINS
FRAUENFELDER, H
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ILLINOIS, BECKMAN INST, URBANA, IL 61801 USA
UNIV ILLINOIS, BECKMAN INST, URBANA, IL 61801 USA
FRAUENFELDER, H
SLIGAR, SG
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ILLINOIS, BECKMAN INST, URBANA, IL 61801 USA
UNIV ILLINOIS, BECKMAN INST, URBANA, IL 61801 USA
SLIGAR, SG
WOLYNES, PG
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ILLINOIS, BECKMAN INST, URBANA, IL 61801 USA
UNIV ILLINOIS, BECKMAN INST, URBANA, IL 61801 USA
WOLYNES, PG
[J].
SCIENCE,
1991,
254
(5038)
: 1598
-
1603
[5]
FRAUENFELDER H, 1988, ANNU REV BIOPHYS BIO, V17, P451
[6]
SELECTIVE ACTIVATION OF INHIBITORY G-PROTEIN ALPHA-SUBUNITS BY PARTIAL AGONISTS OF THE HUMAN 5-HT(1A) RECEPTOR
GETTYS, TW
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV, MED CTR, DEPT MED, DURHAM, NC 27710 USA
GETTYS, TW
FIELDS, TA
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV, MED CTR, DEPT MED, DURHAM, NC 27710 USA
FIELDS, TA
RAYMOND, JR
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV, MED CTR, DEPT MED, DURHAM, NC 27710 USA
RAYMOND, JR
[J].
BIOCHEMISTRY,
1994,
33
(14)
: 4283
-
4290
[7]
AGONIST-RECEPTOR EFFICACY .2. AGONIST TRAFFICKING OF RECEPTOR SIGNALS
KENAKIN, T
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Cellular Biochemistry, Glaxo Research Institute, Research Triangle Park, NC 27709, Five Moore Drive
KENAKIN, T
[J].
TRENDS IN PHARMACOLOGICAL SCIENCES,
1995,
16
(07)
: 232
-
238
[8]
AGONIST-RECEPTOR EFFICACY .1. MECHANISMS OF EFFICACY AND RECEPTOR PROMISCUITY
KENAKIN, T
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Cellular Biochemistry, Glaxo Research Institute, Research Triangle Park, NC 27709, Five Moore Drive
KENAKIN, T
[J].
TRENDS IN PHARMACOLOGICAL SCIENCES,
1995,
16
(06)
: 188
-
192
[9]
AGONIST-SPECIFIC COUPLING OF A CLONED DROSOPHILA OCTOPAMINE TYRAMINE RECEPTOR TO MULTIPLE 2ND MESSENGER SYSTEMS
ROBB, S
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,DEPT ZOOL,AFRC,MOLEC SIGNALLING LAB,CAMBRIDGE CB2 3EJ,ENGLAND
ROBB, S
CHEEK, TR
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,DEPT ZOOL,AFRC,MOLEC SIGNALLING LAB,CAMBRIDGE CB2 3EJ,ENGLAND
CHEEK, TR
HANNAN, FL
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,DEPT ZOOL,AFRC,MOLEC SIGNALLING LAB,CAMBRIDGE CB2 3EJ,ENGLAND
HANNAN, FL
HALL, LM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,DEPT ZOOL,AFRC,MOLEC SIGNALLING LAB,CAMBRIDGE CB2 3EJ,ENGLAND
HALL, LM
MIDGLEY, JM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,DEPT ZOOL,AFRC,MOLEC SIGNALLING LAB,CAMBRIDGE CB2 3EJ,ENGLAND
MIDGLEY, JM
EVANS, PD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,DEPT ZOOL,AFRC,MOLEC SIGNALLING LAB,CAMBRIDGE CB2 3EJ,ENGLAND
EVANS, PD
[J].
EMBO JOURNAL,
1994,
13
(06)
: 1325
-
1330
[10]
SAMAMA P, 1993, J BIOL CHEM, V268, P4625
←
1
2
→