Allosteric modulators of the α7 nicotinic acetylcholine receptor

被引:75
作者
Faghih, Ramin [1 ]
Gopalakrishnan, Murali [1 ]
Briggs, Clark A. [1 ]
机构
[1] Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA
关键词
D O I
10.1021/jm070256g
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:701 / 712
页数:12
相关论文
共 191 条
[51]   α10:: A determinant of nicotinic cholinergic receptor function in mammalian vestibular and cochlear mechanosensory hair cells [J].
Elgoyhen, AB ;
Vetter, DE ;
Katz, E ;
Rothlin, CV ;
Heinemann, SF ;
Boulter, J .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2001, 98 (06) :3501-3506
[52]   Study of the nematode putative GABA type-A receptor subunits: evidence for modulation by ivermectin [J].
Feng, XP ;
Hayashi, J ;
Beech, RN ;
Prichard, RK .
JOURNAL OF NEUROCHEMISTRY, 2002, 83 (04) :870-878
[53]   JN403, in vitro characterization of a novel nicotinic acetylcholine receptor α7 selective agonist [J].
Feuerbach, Dominik ;
Nozulak, Joachim ;
Lingenhoehl, Kurt ;
McAllister, Kevin ;
Hoyer, Daniel .
NEUROSCIENCE LETTERS, 2007, 416 (01) :61-65
[54]   Smoking and Parkinson's and Alzheimer's disease: review of the epidemiological studies [J].
Fratiglioni, L ;
Wang, HX .
BEHAVIOURAL BRAIN RESEARCH, 2000, 113 (1-2) :117-120
[55]  
Frazier CJ, 1998, J NEUROSCI, V18, P1187
[56]  
Gahring Lorise C, 2006, AAPS J, V7, pE885
[57]   Solution NMR of acetylcholine binding protein reveals agonist-mediated conformational change of the C-loop [J].
Gao, Fan ;
Mer, Georges ;
Tonelli, Marco ;
Hansen, Scott B. ;
Burghardt, Thomas P. ;
Taylor, Palmer ;
Sine, Steven M. .
MOLECULAR PHARMACOLOGY, 2006, 70 (04) :1230-1235
[58]   Facilitation of glutamatergic neurotransmission by presynaptic nicotinic acetylcholine receptors [J].
Girod, R ;
Barazangi, N ;
McGehee, D ;
Role, LW .
NEUROPHARMACOLOGY, 2000, 39 (13) :2715-2725
[59]   CELL-SPECIFIC EXPRESSION OF THE ALPHA-9 N-ACH RECEPTOR SUBUNIT IN AUDITORY HAIR-CELLS REVEALED BY SINGLE-CELL RT-PCR [J].
GLOWATZKI, E ;
WILD, K ;
BRANDLE, U ;
FAKLER, G ;
FAKLER, B ;
ZENNER, HP ;
RUPPERSBERG, JP .
PROCEEDINGS OF THE ROYAL SOCIETY B-BIOLOGICAL SCIENCES, 1995, 262 (1364) :141-147
[60]   PHARMACOLOGY AND BIOPHYSICAL PROPERTIES OF ALPHA-7 AND ALPHA-7-ALPHA-8 ALPHA-BUNGAROTOXIN RECEPTOR SUBTYPES IMMUNOPURIFIED FROM THE CHICK OPTIC LOBE [J].
GOTTI, C ;
HANKE, W ;
MAURY, K ;
MORETTI, M ;
BALLIVET, M ;
CLEMENTI, F ;
BERTRAND, D .
EUROPEAN JOURNAL OF NEUROSCIENCE, 1994, 6 (08) :1281-1291