Modular syntheses of isoxazoloazepinones and pyrazoloazepinones

被引：38

作者：

Adamo, Mauro F. A.

Duffy, Eleanor F.

Donati, Donato

Sarti-Fantoni, Piero

机构：

[1] Royal Coll Surgeons Ireland, Dept Pharmaceut & Med Chem, CSCB, Dublin 2, Ireland

[2] Univ Siena, Dipartimento Chim, I-53100 Siena, Italy

[3] Univ Florence, Dipartimento Chim Organ U Schiff, I-50019 Sesto Fiorentino, Italy

来源：

TETRAHEDRON | 2007年 / 63卷 / 12期

关键词：

fused isoxazoles; polyfunctional scaffold; fused pyrazoles;

D O I：

10.1016/j.tet.2007.01.018

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Herein we described an optimised synthesis of isoxazoloazepi none and novel heterocycle pyrazoloazepinone. These syntheses are modular in nature and fast to execute. The title compounds were obtained pure without the intervention of chromatography. (c) 2007 Elsevier Ltd. All rights reserved.

引用

收藏

页码：2684 / 2688

页数：5

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