Design of remarkably simple, yet potent urea-based inhibitors of glutamate carboxypeptidase II (NAALADase)

被引:211
作者
Kozikowski, AP
Nan, F
Conti, P
Zhang, JH
Ramadan, E
Bzdega, T
Wroblewska, B
Neale, JH
Pshenichkin, S
Wroblewski, JT
机构
[1] Georgetown Univ, Med Ctr, Drug Discovery Program, Dept Neurol, Washington, DC 20007 USA
[2] Georgetown Univ, Med Ctr, Dept Pharmacol, Washington, DC 20007 USA
[3] Georgetown Univ, Dept Biol, Washington, DC 20057 USA
关键词
D O I
10.1021/jm000406m
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:298 / 301
页数:4
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