A simple and new method for the synthesis of 1,5-benzodiazepine derivatives on a solid surface

被引：219

作者：

Balakrishna, MS ^{[1
]}

Kaboudin, B

机构：

[1] Indian Inst Technol, Dept Chem, Bombay 400076, Maharashtra, India

[2] IASBS, Gava Zang 45195, Zanjan, Iran

来源：

TETRAHEDRON LETTERS | 2001年 / 42卷 / 06期

关键词：

benzodiazepine; magnesium oxide; phosphorus oxychloride; ketones;

D O I：

10.1016/S0040-4039(00)02168-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Magnesium oxide/phosphorus oxychloride (MOPO) was found to be an efficient reagent for the preparation of 1,5-benzodiazepine derivatives of o-phenylenediamine and ketones. This method is an easy, rapid, and high yielding reaction for the synthesis of 1,5-benzodiazepine derivatives. (C) 2001 Elsevier Science Ltd. All rights reserved.

引用

页码：1127 / 1129

页数：3

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