Synthesis of chiral pyrazoles and isoxazoles as constrained amino acids

被引：38

作者：

Falorni, M ^{[1
]}

Giacomelli, G ^{[1
]}

Spanedda, AM ^{[1
]}

机构：

[1] Univ Sassari, Dipartimento Chim, I-07100 Sassari, Italy

来源：

TETRAHEDRON-ASYMMETRY | 1998年 / 9卷 / 17期

关键词：

D O I：

10.1016/S0957-4166(98)00305-X

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

A stereospecific syntheses of optically active pyrazoles and isoxazoles from L-proline is described. The procedure presented is based on readily available materials and can be used for preparing new conformationally restricted pyrazole-containing amino acids, (C) 1998 Elsevier Science Ltd. All rights reserved.

引用

页码：3039 / 3046

页数：8

共 13 条

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