Synthesis of new oxazole-containing peptidomimetics

被引：25

作者：

Falorni, M ^{[1
]}

Dettori, G ^{[1
]}

Giacomelli, G ^{[1
]}

机构：

[1] Univ Sassari, Dipartimento Chim, I-07100 Sassari, Italy

来源：

TETRAHEDRON-ASYMMETRY | 1998年 / 9卷 / 08期

关键词：

D O I：

10.1016/S0957-4166(98)00109-8

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

Enantiospecific syntheses of optically active amino acids containing an oxazole moiety are described. Two different strategies for their insertion in a peptidomimetic chain are also discussed. The procedures presented are based on materials readily available in multigram quantities. (C) 1998 Elsevier Science Ltd. All rights reserved.

引用

页码：1419 / 1426

页数：8

共 18 条

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