Targeting Bcl-2 and Bcl-XL with nonpeptidic small-molecule antagonists

被引:127
作者
Wang, SM
Yang, DJ
Lippman, ME
机构
[1] Univ Michigan, Sch Med, Dept Internal Med, Taubman Ctr 3101, Ann Arbor, MI 48109 USA
[2] Univ Michigan, Sch Med, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA
关键词
D O I
10.1053/j.seminoncol.2003.08.015
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:133 / 142
页数:10
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共 66 条
[21]  
Leech SH, 2000, INT J CANCER, V86, P570, DOI 10.1002/(SICI)1097-0215(20000515)86:4<570::AID-IJC20>3.3.CO
[22]  
2-K
[23]   Antiapoptotic bcl-2 and bcl-xL in advanced malignant melanoma [J].
Leiter, U ;
Schmid, RM ;
Kaskel, P ;
Peter, RU ;
Krähn, G .
ARCHIVES OF DERMATOLOGICAL RESEARCH, 2000, 292 (05) :225-232
[24]   Distinct BH3 domains either sensitize or activate mitochondrial apoptosis, serving as prototype cancer therapeutics [J].
Letai, A ;
Bassik, MC ;
Walensky, LD ;
Sorcinelli, MD ;
Weiler, S ;
Korsmeyer, SJ .
CANCER CELL, 2002, 2 (03) :183-192
[25]  
Makino S, 1997, J COMPUT CHEM, V18, P1812, DOI 10.1002/(SICI)1096-987X(19971115)18:14<1812::AID-JCC10>3.0.CO
[26]  
2-H
[27]  
Manne U, 1997, INT J CANCER, V74, P346, DOI 10.1002/(SICI)1097-0215(19970620)74:3<346::AID-IJC19>3.0.CO
[28]  
2-9
[29]   Apoptosis inhibiting factor Bcl-xL might be the crucial member of the Bcl-2 gene family in colorectal cancer [J].
Maurer, CA ;
Friess, H ;
Bühler, SS ;
Wahl, BR ;
Graber, H ;
Zimmermann, A ;
Büchler, MW .
DIGESTIVE DISEASES AND SCIENCES, 1998, 43 (12) :2641-2648
[30]  
MICHAEL S, 1997, SCIENCE, V275, P983