Endothelin antagonists

被引:32
作者
Lago, MA [1 ]
Luengo, JI [1 ]
Peishoff, CE [1 ]
Elliott, JD [1 ]
机构
[1] SMITHKLINE BEECHAM PHARMACEUT PLC, KING OF PRUSSIA, PA 19406 USA
来源
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 31 | 1996年 / 31卷
关键词
D O I
10.1016/S0065-7743(08)60448-0
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:81 / 90
页数:10
相关论文
共 73 条
[1]  
[Anonymous], 1995, J CARDIOVASC PHAR S3, V26, pS1
[2]  
ASTLES PC, 1995, 8 SCI RSC MED CHEM S
[3]   INTERACTION OF ENDOTHELIN-3 WITH ENDOTHELIN-B RECEPTOR IS ESSENTIAL FOR DEVELOPMENT OF EPIDERMAL MELANOCYTES AND ENTERIC NEURONS [J].
BAYNASH, AG ;
HOSODA, K ;
GIAID, A ;
RICHARDSON, JA ;
EMOTO, N ;
HAMMER, RE ;
YANAGISAWA, M .
CELL, 1994, 79 (07) :1277-1285
[4]  
BENNETT T, 1994, J HUM HYPERTENS, V8, P587
[5]   PHOSPHORUS-CONTAINING INHIBITORS OF ENDOTHELIN CONVERTING ENZYME - EFFECTS OF THE ELECTRONIC NATURE OF PHOSPHORUS ON INHIBITOR POTENCY [J].
BERTENSHAW, SR ;
ROGERS, RS ;
STERN, MK ;
NORMAN, BH ;
MOORE, WM ;
JEROME, GM ;
BRANSON, LM ;
MCDONALD, JF ;
MCMAHON, EG ;
PALOMO, MA .
JOURNAL OF MEDICINAL CHEMISTRY, 1993, 36 (01) :173-176
[6]   THIOL AND HYDROXAMIC ACID-CONTAINING INHIBITORS OF ENDOTHELIN-CONVERTING ENZYME [J].
BERTENSHAW, SR ;
TALLEY, JJ ;
ROGERS, RS ;
CARTER, JS ;
MOORE, WM ;
BRANSON, LM ;
KOBOLDT, CM .
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1993, 3 (10) :1953-1958
[7]  
BIALECKI R, 1996, ENDOTHELIN INHIBITOR
[8]   HYDROXAMIC ACIDS AS POTENT INHIBITORS OF ENDOTHELIN-CONVERTING ENZYME FROM HUMAN BRONCHIOLAR SMOOTH-MUSCLE [J].
BIHOVSKY, R ;
LEVINSON, BL ;
LOEWI, RC ;
ERHARDT, PW ;
POLOKOFF, MA .
JOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (12) :2119-2129
[9]  
BROCK TA, 1996, ENDOTHELIN INHIBITOR
[10]   Blockade of radiocontrast-induced nephrotoxicity by the endothelin receptor antagonist, SB 209670 [J].
Brooks, DP ;
DePalma, PD .
NEPHRON, 1996, 72 (04) :629-636