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DNA gyrase as a drug target
被引:95
作者
:
Maxwell, A
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Leicester, Dept Biochem, Leicester LE1 7RH, Leics, England
Univ Leicester, Dept Biochem, Leicester LE1 7RH, Leics, England
Maxwell, A
[
1
]
机构
:
[1]
Univ Leicester, Dept Biochem, Leicester LE1 7RH, Leics, England
来源
:
BIOCHEMICAL SOCIETY TRANSACTIONS
|
1999年
/ 27卷
/ 02期
基金
:
英国惠康基金;
关键词
:
D O I
:
10.1042/bst0270048
中图分类号
:
Q5 [生物化学];
Q7 [分子生物学];
学科分类号
:
071010 ;
081704 ;
摘要
:
引用
收藏
页码:48 / 53
页数:6
相关论文
共 34 条
[1]
THE 43-KILODALTON N-TERMINAL FRAGMENT OF THE DNA GYRASE-B PROTEIN HYDROLYZES ATP AND BINDS COUMARIN DRUGS
ALI, JA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
ALI, JA
JACKSON, AP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
JACKSON, AP
HOWELLS, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
HOWELLS, AJ
MAXWELL, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
MAXWELL, A
[J].
BIOCHEMISTRY,
1993,
32
(10)
: 2717
-
2724
[2]
Bates A. D., 1993, DNA topology
[3]
Crystal structure of the breakage-reunion domain of DNA gyrase
Cabral, JHM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
Cabral, JHM
Jackson, AP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
Jackson, AP
Smith, CV
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
Smith, CV
Shikotra, N
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
Shikotra, N
Maxwell, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
Maxwell, A
Liddington, RC
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
Liddington, RC
[J].
NATURE,
1997,
388
(6645)
: 903
-
906
[4]
LOCAL SEQUENCE REQUIREMENTS FOR DNA CLEAVAGE BY MAMMALIAN TOPOISOMERASE-II IN THE PRESENCE OF DOXORUBICIN
CAPRANICO, G
论文数:
0
引用数:
0
h-index:
0
机构:
NCI,DIV CANC TREATMENT,MOLEC PHARMACOL LAB,BETHESDA,MD 20892
NCI,DIV CANC TREATMENT,MOLEC PHARMACOL LAB,BETHESDA,MD 20892
CAPRANICO, G
KOHN, KW
论文数:
0
引用数:
0
h-index:
0
机构:
NCI,DIV CANC TREATMENT,MOLEC PHARMACOL LAB,BETHESDA,MD 20892
NCI,DIV CANC TREATMENT,MOLEC PHARMACOL LAB,BETHESDA,MD 20892
KOHN, KW
POMMIER, Y
论文数:
0
引用数:
0
h-index:
0
机构:
NCI,DIV CANC TREATMENT,MOLEC PHARMACOL LAB,BETHESDA,MD 20892
NCI,DIV CANC TREATMENT,MOLEC PHARMACOL LAB,BETHESDA,MD 20892
POMMIER, Y
[J].
NUCLEIC ACIDS RESEARCH,
1990,
18
(22)
: 6611
-
6619
[5]
CONTRERAS A, 1992, MOL MICROBIOL, V6, P1617
[6]
DNA cleavage is not required for the binding of quinolone drugs to the DNA Gyrase - DNA complex
Critchlow, SE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER,DEPT BIOCHEM,LEICESTER LE1 7RH,LEICS,ENGLAND
UNIV LEICESTER,DEPT BIOCHEM,LEICESTER LE1 7RH,LEICS,ENGLAND
Critchlow, SE
Maxwell, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER,DEPT BIOCHEM,LEICESTER LE1 7RH,LEICS,ENGLAND
UNIV LEICESTER,DEPT BIOCHEM,LEICESTER LE1 7RH,LEICS,ENGLAND
Maxwell, A
[J].
BIOCHEMISTRY,
1996,
35
(23)
: 7387
-
7393
[7]
DNA gyrase, topoisomerase IV, and the 4-quinolones
Drlica, K
论文数:
0
引用数:
0
h-index:
0
机构:
Public Health Research Institute, New York
Drlica, K
Zhao, XL
论文数:
0
引用数:
0
h-index:
0
机构:
Public Health Research Institute, New York
Zhao, XL
[J].
MICROBIOLOGY AND MOLECULAR BIOLOGY REVIEWS,
1997,
61
(03)
: 377
-
+
[8]
DIFFERENTIAL-EFFECTS OF ANTIBIOTICS INHIBITING GYRASE
ENGLE, EC
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ROCHESTER,DEPT BIOL,ROCHESTER,NY 14627
UNIV ROCHESTER,DEPT BIOL,ROCHESTER,NY 14627
ENGLE, EC
MANES, SH
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ROCHESTER,DEPT BIOL,ROCHESTER,NY 14627
UNIV ROCHESTER,DEPT BIOL,ROCHESTER,NY 14627
MANES, SH
DRLICA, K
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ROCHESTER,DEPT BIOL,ROCHESTER,NY 14627
UNIV ROCHESTER,DEPT BIOL,ROCHESTER,NY 14627
DRLICA, K
[J].
JOURNAL OF BACTERIOLOGY,
1982,
149
(01)
: 92
-
98
[9]
EVERETT MJ, 1997, HDB PHARM QUINOLONE, P259
[10]
MUTATIONAL ANALYSIS OF A TYPE-II TOPOISOMERASE CLEAVAGE SITE - DISTINCT REQUIREMENTS FOR ENZYME AND INHIBITORS
FREUDENREICH, CH
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,MED CTR,DEPT MICROBIOL & IMMUNOL,DURHAM,NC 27710
DUKE UNIV,MED CTR,DEPT MICROBIOL & IMMUNOL,DURHAM,NC 27710
FREUDENREICH, CH
KREUZER, KN
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,MED CTR,DEPT MICROBIOL & IMMUNOL,DURHAM,NC 27710
DUKE UNIV,MED CTR,DEPT MICROBIOL & IMMUNOL,DURHAM,NC 27710
KREUZER, KN
[J].
EMBO JOURNAL,
1993,
12
(05)
: 2085
-
2097
←
1
2
3
4
→
共 34 条
[1]
THE 43-KILODALTON N-TERMINAL FRAGMENT OF THE DNA GYRASE-B PROTEIN HYDROLYZES ATP AND BINDS COUMARIN DRUGS
ALI, JA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
ALI, JA
JACKSON, AP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
JACKSON, AP
HOWELLS, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
HOWELLS, AJ
MAXWELL, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
UNIV LEICESTER,DEPT BIOCHEM,UNIV RD,LEICESTER LE1 7RH,ENGLAND
MAXWELL, A
[J].
BIOCHEMISTRY,
1993,
32
(10)
: 2717
-
2724
[2]
Bates A. D., 1993, DNA topology
[3]
Crystal structure of the breakage-reunion domain of DNA gyrase
Cabral, JHM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
Cabral, JHM
Jackson, AP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
Jackson, AP
Smith, CV
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
Smith, CV
Shikotra, N
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
Shikotra, N
Maxwell, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
Maxwell, A
Liddington, RC
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
UNIV LEICESTER, DEPT BIOCHEM, LEICESTER LE1 7RH, LEICS, ENGLAND
Liddington, RC
[J].
NATURE,
1997,
388
(6645)
: 903
-
906
[4]
LOCAL SEQUENCE REQUIREMENTS FOR DNA CLEAVAGE BY MAMMALIAN TOPOISOMERASE-II IN THE PRESENCE OF DOXORUBICIN
CAPRANICO, G
论文数:
0
引用数:
0
h-index:
0
机构:
NCI,DIV CANC TREATMENT,MOLEC PHARMACOL LAB,BETHESDA,MD 20892
NCI,DIV CANC TREATMENT,MOLEC PHARMACOL LAB,BETHESDA,MD 20892
CAPRANICO, G
KOHN, KW
论文数:
0
引用数:
0
h-index:
0
机构:
NCI,DIV CANC TREATMENT,MOLEC PHARMACOL LAB,BETHESDA,MD 20892
NCI,DIV CANC TREATMENT,MOLEC PHARMACOL LAB,BETHESDA,MD 20892
KOHN, KW
POMMIER, Y
论文数:
0
引用数:
0
h-index:
0
机构:
NCI,DIV CANC TREATMENT,MOLEC PHARMACOL LAB,BETHESDA,MD 20892
NCI,DIV CANC TREATMENT,MOLEC PHARMACOL LAB,BETHESDA,MD 20892
POMMIER, Y
[J].
NUCLEIC ACIDS RESEARCH,
1990,
18
(22)
: 6611
-
6619
[5]
CONTRERAS A, 1992, MOL MICROBIOL, V6, P1617
[6]
DNA cleavage is not required for the binding of quinolone drugs to the DNA Gyrase - DNA complex
Critchlow, SE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER,DEPT BIOCHEM,LEICESTER LE1 7RH,LEICS,ENGLAND
UNIV LEICESTER,DEPT BIOCHEM,LEICESTER LE1 7RH,LEICS,ENGLAND
Critchlow, SE
Maxwell, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LEICESTER,DEPT BIOCHEM,LEICESTER LE1 7RH,LEICS,ENGLAND
UNIV LEICESTER,DEPT BIOCHEM,LEICESTER LE1 7RH,LEICS,ENGLAND
Maxwell, A
[J].
BIOCHEMISTRY,
1996,
35
(23)
: 7387
-
7393
[7]
DNA gyrase, topoisomerase IV, and the 4-quinolones
Drlica, K
论文数:
0
引用数:
0
h-index:
0
机构:
Public Health Research Institute, New York
Drlica, K
Zhao, XL
论文数:
0
引用数:
0
h-index:
0
机构:
Public Health Research Institute, New York
Zhao, XL
[J].
MICROBIOLOGY AND MOLECULAR BIOLOGY REVIEWS,
1997,
61
(03)
: 377
-
+
[8]
DIFFERENTIAL-EFFECTS OF ANTIBIOTICS INHIBITING GYRASE
ENGLE, EC
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ROCHESTER,DEPT BIOL,ROCHESTER,NY 14627
UNIV ROCHESTER,DEPT BIOL,ROCHESTER,NY 14627
ENGLE, EC
MANES, SH
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ROCHESTER,DEPT BIOL,ROCHESTER,NY 14627
UNIV ROCHESTER,DEPT BIOL,ROCHESTER,NY 14627
MANES, SH
DRLICA, K
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ROCHESTER,DEPT BIOL,ROCHESTER,NY 14627
UNIV ROCHESTER,DEPT BIOL,ROCHESTER,NY 14627
DRLICA, K
[J].
JOURNAL OF BACTERIOLOGY,
1982,
149
(01)
: 92
-
98
[9]
EVERETT MJ, 1997, HDB PHARM QUINOLONE, P259
[10]
MUTATIONAL ANALYSIS OF A TYPE-II TOPOISOMERASE CLEAVAGE SITE - DISTINCT REQUIREMENTS FOR ENZYME AND INHIBITORS
FREUDENREICH, CH
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,MED CTR,DEPT MICROBIOL & IMMUNOL,DURHAM,NC 27710
DUKE UNIV,MED CTR,DEPT MICROBIOL & IMMUNOL,DURHAM,NC 27710
FREUDENREICH, CH
KREUZER, KN
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,MED CTR,DEPT MICROBIOL & IMMUNOL,DURHAM,NC 27710
DUKE UNIV,MED CTR,DEPT MICROBIOL & IMMUNOL,DURHAM,NC 27710
KREUZER, KN
[J].
EMBO JOURNAL,
1993,
12
(05)
: 2085
-
2097
←
1
2
3
4
→