Preparation of (S)-3-carbethoxy-3-benzylpiperidine and the growth hormone secretagogue L-163,540

被引：9

作者：

Maligres, PE

Chartrain, MM

Upadhyay, V

Cohen, D

Reamer, RA

Askin, D

Volante, RP

Reider, PJ

机构：

[1] Merck & Co Inc, Merck Res Labs, Dept Proc Res, Rahway, NJ 07065 USA

[2] Merck & Co Inc, Merck Res Labs, Dept Bioproc Res, Rahway, NJ 07065 USA

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1998年 / 63卷 / 25期

关键词：

D O I：

10.1021/jo980990v

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[No abstract available]

引用

页码：9548 / 9551

页数：4

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[6] A NONPEPTIDYL GROWTH-HORMONE SECRETAGOGUE [J].

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[7] 1-[2(R)-(2-amino-2-methylpropionylamino)-3-(1H-indol-3-yl)propionyl]-3-benzylpiperidine-3(S)-carboxylic acid ethyl ester (L-163,540):: A potent, orally bioavailable, and short-duration growth hormone secretagogue [J].

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