The discovery of ezetimibe: A view from outside the receptor

[1] Effect of ezetimibe coadministered with atorvastatin in 628 patients with primary hypercholesterolemia - A prospective, randomized, double-blind trial [J]. CIRCULATION, 2003, 107 (19) : 2409 - 2415

[2] Ezetimibe [J]. EXPERT OPINION ON INVESTIGATIONAL DRUGS, 2002, 11 (11) : 1587 - 1604

[3] New lipid-modifying therapies [J]. EXPERT OPINION ON INVESTIGATIONAL DRUGS, 2003, 12 (03) : 325 - 335

[4] 2-AZETIDINONES AS INHIBITORS OF CHOLESTEROL ABSORPTION [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1994, 37 (12) : 1733 - 1736

[5] ASYMMETRIC-SYNTHESIS AND ABSOLUTE STEREOCHEMISTRY OF CHOLESTEROL ABSORPTION INHIBITOR, SCH-48461 [J]. TETRAHEDRON LETTERS, 1994, 35 (40) : 7339 - 7342

[6] BURNETT DA, IN PRESS CURR TOP ME

[7] SUBSTITUTED (1,2-DIARYLETHYL)AMIDE ACYL-COA-CHOLESTEROL ACYLTRANSFERASE INHIBITORS - EFFECT OF POLAR GROUPS ON IN-VITRO AND IN-VIVO ACTIVITY [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (10) : 1600 - 1607

[8] 2-azetidinone cholesterol absorption inhibitors: Structure-activity relationships on the heterocyclic nucleus [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1996, 39 (19) : 3684 - 3693

[9] DESIGN OF POTENT COMPETITIVE INHIBITORS OF ANGIOTENSIN-CONVERTING ENZYME - CARBOXYALKANOYL AND MERCAPTOALKANOYL AMINO-ACIDS [J]. BIOCHEMISTRY, 1977, 16 (25) : 5484 - 5491

[10] Ezetimibe [J]. American Journal of Cardiovascular Drugs, 2003, 3 (1) : 67 - 76

[1] Effect of ezetimibe coadministered with atorvastatin in 628 patients with primary hypercholesterolemia - A prospective, randomized, double-blind trial [J]. CIRCULATION, 2003, 107 (19) : 2409 - 2415

[2] Ezetimibe [J]. EXPERT OPINION ON INVESTIGATIONAL DRUGS, 2002, 11 (11) : 1587 - 1604

[3] New lipid-modifying therapies [J]. EXPERT OPINION ON INVESTIGATIONAL DRUGS, 2003, 12 (03) : 325 - 335

[4] 2-AZETIDINONES AS INHIBITORS OF CHOLESTEROL ABSORPTION [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1994, 37 (12) : 1733 - 1736

[5] ASYMMETRIC-SYNTHESIS AND ABSOLUTE STEREOCHEMISTRY OF CHOLESTEROL ABSORPTION INHIBITOR, SCH-48461 [J]. TETRAHEDRON LETTERS, 1994, 35 (40) : 7339 - 7342

[6] BURNETT DA, IN PRESS CURR TOP ME

[7] SUBSTITUTED (1,2-DIARYLETHYL)AMIDE ACYL-COA-CHOLESTEROL ACYLTRANSFERASE INHIBITORS - EFFECT OF POLAR GROUPS ON IN-VITRO AND IN-VIVO ACTIVITY [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (10) : 1600 - 1607

[8] 2-azetidinone cholesterol absorption inhibitors: Structure-activity relationships on the heterocyclic nucleus [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1996, 39 (19) : 3684 - 3693

[9] DESIGN OF POTENT COMPETITIVE INHIBITORS OF ANGIOTENSIN-CONVERTING ENZYME - CARBOXYALKANOYL AND MERCAPTOALKANOYL AMINO-ACIDS [J]. BIOCHEMISTRY, 1977, 16 (25) : 5484 - 5491

[10] Ezetimibe [J]. American Journal of Cardiovascular Drugs, 2003, 3 (1) : 67 - 76