A versatile one-pot synthesis of 4-aryl-1,5-disubstituted 1,2,3-triazoles via 1,3-dipolar cycloaddition followed by Negishi reaction under new conditions

被引：24

作者：

Akao, Atsushi

Tsuritani, Takayuki

Kii, Satoshi

Sato, Kimihiko

Nonoyama, Nobuaki

Mase, Toshiaki

Yasuda, Nobuyoshi

机构：

[1] Merck Res Labs, Tsukuba, Ibaraki 3002611, Japan

[2] Merck Res Labs, Dept Proc Res, Rahway, NJ 07065 USA

来源：

SYNLETT | 2007年 / 01期

关键词：

triazole; Negishi reaction; 1,3-dipolar cycloaddition; XANTPHOS; zinc; cross-coupling;

D O I：

10.1055/s-2006-958435

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Several derivatives of 4-aryl-1,5-disubstituted 1,2,3-triazole were synthesized in good yields via 1,3-dipolar cycloaddition followed by Negishi reaction under new conditions.

引用

页码：31 / 36

页数：6

共 61 条

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