Protein delivery from poly(lactic-co-glycolic acid) biodegradable microspheres: release kinetics and stability issues

被引:227
作者
Crotts, G
Park, TG [1 ]
机构
[1] Korea Adv Inst Sci & Technol, Dept Biol Sci, Taejon 305701, South Korea
[2] Warner Lambert Parke Davis, Pharmaceut Delivery Syst R&D, Morris Plains, NJ 07950 USA
关键词
protein delivery; biodegradable; PLGA; stability; release kinetics; microsphere;
D O I
10.3109/02652049809008253
中图分类号
O69 [应用化学];
学科分类号
081704 [应用化学];
摘要
引用
收藏
页码:699 / 713
页数:15
相关论文
共 28 条
[1]
DETERMINANTS OF RELEASE RATE OF TETANUS VACCINE FROM POLYESTER MICROSPHERES [J].
ALONSO, MJ ;
COHEN, S ;
PARK, TG ;
GUPTA, RK ;
SIBER, GR ;
LANGER, R .
PHARMACEUTICAL RESEARCH, 1993, 10 (07) :945-953
[2]
CLELAND JL, 1994, ACS SYM SER, V567, P1
[3]
CONTROLLED DELIVERY SYSTEMS FOR PROTEINS BASED ON POLY(LACTIC GLYCOLIC ACID) MICROSPHERES [J].
COHEN, S ;
YOSHIOKA, T ;
LUCARELLI, M ;
HWANG, LH ;
LANGER, R .
PHARMACEUTICAL RESEARCH, 1991, 8 (06) :713-720
[4]
PREPARATION OF POROUS AND NONPOROUS BIODEGRADABLE POLYMERIC HOLLOW MICROSPHERES [J].
CROTTS, G ;
PARK, TG .
JOURNAL OF CONTROLLED RELEASE, 1995, 35 (2-3) :91-105
[5]
Stability and release of bovine serum albumin encapsulated within poly(D,L-lactide-co-glycolide) microparticles [J].
Crotts, G ;
Park, TG .
JOURNAL OF CONTROLLED RELEASE, 1997, 44 (2-3) :123-134
[6]
Adsorption determines in-vitro protein release rate from biodegradable microspheres: Quantitative analysis of surface area during degradation [J].
Crotts, G ;
Sah, H ;
Park, TG .
JOURNAL OF CONTROLLED RELEASE, 1997, 47 (01) :101-111
[7]
CURKE PA, 1996, P INT S CONTR REL BI, V23, P133
[8]
RELEASE OF HUMAN SERUM-ALBUMIN FROM POLY(LACTIDE-CO-GLYCOLIDE) MICROSPHERES [J].
HORA, MS ;
RANA, RK ;
NUNBERG, JH ;
TICE, TR ;
GILLEY, RM ;
HUDSON, ME .
PHARMACEUTICAL RESEARCH, 1990, 7 (11) :1190-1194
[9]
BIODEGRADABLE POLYMER SYSTEMS FOR THE SUSTAINED-RELEASE OF POLYPEPTIDES [J].
HUTCHINSON, FG ;
FURR, BJA .
JOURNAL OF CONTROLLED RELEASE, 1990, 13 (2-3) :279-294
[10]
THE PREPARATION AND CHARACTERIZATION OF POLY(LACTIDE-CO-GLYCOLIDE) MICROPARTICLES .2. THE ENTRAPMENT OF A MODEL PROTEIN USING A (WATER-IN-OIL)-IN-WATER EMULSION SOLVENT EVAPORATION TECHNIQUE [J].
JEFFERY, H ;
DAVIS, SS ;
OHAGAN, DT .
PHARMACEUTICAL RESEARCH, 1993, 10 (03) :362-368