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Binding of an inhibitor of the p53/MDM2 interaction to MDM2
被引:57
作者
:
Duncan, SJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Dept Chem, Cambridge CB2 1EW, England
Univ Cambridge, Dept Chem, Cambridge CB2 1EW, England
Duncan, SJ
[
1
]
Cooper, MA
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Dept Chem, Cambridge CB2 1EW, England
Univ Cambridge, Dept Chem, Cambridge CB2 1EW, England
Cooper, MA
[
1
]
Williams, DH
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Dept Chem, Cambridge CB2 1EW, England
Univ Cambridge, Dept Chem, Cambridge CB2 1EW, England
Williams, DH
[
1
]
机构
:
[1]
Univ Cambridge, Dept Chem, Cambridge CB2 1EW, England
来源
:
CHEMICAL COMMUNICATIONS
|
2003年
/ 03期
关键词
:
D O I
:
10.1039/b211889k
中图分类号
:
O6 [化学];
学科分类号
:
0703 ;
摘要
:
The mode of action of the secondary metabolite chlorofusin, which antagonises the interaction between p53 and MDM2, involves direct binding to the N-terminal domain of MDM2.
引用
收藏
页码:316 / 317
页数:2
相关论文
共 10 条
[1]
On the interaction between p53 and MDM2: Transfer NOE study of a p53-derived peptide ligated to MDM2
Blommers, MJJ
论文数:
0
引用数:
0
h-index:
0
机构:
Physics, Core Drug Discovery Technologies, Ciba-Geigy AG, CH-4002 Basel, P.O. Box
Blommers, MJJ
Fendrich, G
论文数:
0
引用数:
0
h-index:
0
机构:
Physics, Core Drug Discovery Technologies, Ciba-Geigy AG, CH-4002 Basel, P.O. Box
Fendrich, G
GarciaEcheverria, C
论文数:
0
引用数:
0
h-index:
0
机构:
Physics, Core Drug Discovery Technologies, Ciba-Geigy AG, CH-4002 Basel, P.O. Box
GarciaEcheverria, C
Chene, P
论文数:
0
引用数:
0
h-index:
0
机构:
Physics, Core Drug Discovery Technologies, Ciba-Geigy AG, CH-4002 Basel, P.O. Box
Chene, P
[J].
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-
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[2]
BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3
[3]
Bacillus thuringiensis Cry1Ac toxin interaction with Manduca sexta aminopeptidase N in a model membrane environment
Cooper, MA
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Dept Biochem, Cambridge CB2 1GA, England
Cooper, MA
Carroll, J
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引用数:
0
h-index:
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机构:
Univ Cambridge, Dept Biochem, Cambridge CB2 1GA, England
Carroll, J
Travis, ER
论文数:
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引用数:
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h-index:
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机构:
Univ Cambridge, Dept Biochem, Cambridge CB2 1GA, England
Travis, ER
Williams, DH
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Dept Biochem, Cambridge CB2 1GA, England
Williams, DH
Ellar, DJ
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0
引用数:
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0
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Univ Cambridge, Dept Biochem, Cambridge CB2 1GA, England
Univ Cambridge, Dept Biochem, Cambridge CB2 1GA, England
Ellar, DJ
[J].
BIOCHEMICAL JOURNAL,
1998,
333
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683
[4]
Isolation and structure elucidation of chlorofusin, a novel p53-MDM2 antagonist from a Fusarium sp.
Duncan, SJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Duncan, SJ
Grüschow, S
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Grüschow, S
Williams, DH
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Williams, DH
McNicholas, C
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
McNicholas, C
Purewal, R
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Purewal, R
Hajek, M
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Hajek, M
Gerlitz, M
论文数:
0
引用数:
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h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Gerlitz, M
Martin, S
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0
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Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Martin, S
Wrigley, SK
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Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
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Moore, M
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Kussie, PH
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MEM SLOAN KETTERING CANC CTR,CELLULAR BIOCHEM & BIOPHYS PROGRAM,NEW YORK,NY 10021
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共 10 条
[1]
On the interaction between p53 and MDM2: Transfer NOE study of a p53-derived peptide ligated to MDM2
Blommers, MJJ
论文数:
0
引用数:
0
h-index:
0
机构:
Physics, Core Drug Discovery Technologies, Ciba-Geigy AG, CH-4002 Basel, P.O. Box
Blommers, MJJ
Fendrich, G
论文数:
0
引用数:
0
h-index:
0
机构:
Physics, Core Drug Discovery Technologies, Ciba-Geigy AG, CH-4002 Basel, P.O. Box
Fendrich, G
GarciaEcheverria, C
论文数:
0
引用数:
0
h-index:
0
机构:
Physics, Core Drug Discovery Technologies, Ciba-Geigy AG, CH-4002 Basel, P.O. Box
GarciaEcheverria, C
Chene, P
论文数:
0
引用数:
0
h-index:
0
机构:
Physics, Core Drug Discovery Technologies, Ciba-Geigy AG, CH-4002 Basel, P.O. Box
Chene, P
[J].
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1997,
119
(14)
: 3425
-
3426
[2]
BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3
[3]
Bacillus thuringiensis Cry1Ac toxin interaction with Manduca sexta aminopeptidase N in a model membrane environment
Cooper, MA
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Dept Biochem, Cambridge CB2 1GA, England
Cooper, MA
Carroll, J
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Dept Biochem, Cambridge CB2 1GA, England
Carroll, J
Travis, ER
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Dept Biochem, Cambridge CB2 1GA, England
Travis, ER
Williams, DH
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Dept Biochem, Cambridge CB2 1GA, England
Williams, DH
Ellar, DJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Dept Biochem, Cambridge CB2 1GA, England
Univ Cambridge, Dept Biochem, Cambridge CB2 1GA, England
Ellar, DJ
[J].
BIOCHEMICAL JOURNAL,
1998,
333
: 677
-
683
[4]
Isolation and structure elucidation of chlorofusin, a novel p53-MDM2 antagonist from a Fusarium sp.
Duncan, SJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Duncan, SJ
Grüschow, S
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Grüschow, S
Williams, DH
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Williams, DH
McNicholas, C
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
McNicholas, C
Purewal, R
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Purewal, R
Hajek, M
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Hajek, M
Gerlitz, M
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Gerlitz, M
Martin, S
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Martin, S
Wrigley, SK
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Wrigley, SK
Moore, M
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Univ Cambridge, Cambridge Ctr Mol Recognit, Chem Lab, Cambridge CB2 1EW, England
Moore, M
[J].
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
2001,
123
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: 554
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560
[5]
Structure of the MDM2 oncoprotein bound to the p53 tumor suppressor transactivation domain
Kussie, PH
论文数:
0
引用数:
0
h-index:
0
机构:
MEM SLOAN KETTERING CANC CTR,CELLULAR BIOCHEM & BIOPHYS PROGRAM,NEW YORK,NY 10021
Kussie, PH
Gorina, S
论文数:
0
引用数:
0
h-index:
0
机构:
MEM SLOAN KETTERING CANC CTR,CELLULAR BIOCHEM & BIOPHYS PROGRAM,NEW YORK,NY 10021
Gorina, S
Marechal, V
论文数:
0
引用数:
0
h-index:
0
机构:
MEM SLOAN KETTERING CANC CTR,CELLULAR BIOCHEM & BIOPHYS PROGRAM,NEW YORK,NY 10021
Marechal, V
Elenbaas, B
论文数:
0
引用数:
0
h-index:
0
机构:
MEM SLOAN KETTERING CANC CTR,CELLULAR BIOCHEM & BIOPHYS PROGRAM,NEW YORK,NY 10021
Elenbaas, B
Moreau, J
论文数:
0
引用数:
0
h-index:
0
机构:
MEM SLOAN KETTERING CANC CTR,CELLULAR BIOCHEM & BIOPHYS PROGRAM,NEW YORK,NY 10021
Moreau, J
Levine, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
MEM SLOAN KETTERING CANC CTR,CELLULAR BIOCHEM & BIOPHYS PROGRAM,NEW YORK,NY 10021
Levine, AJ
Pavletich, NP
论文数:
0
引用数:
0
h-index:
0
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MEM SLOAN KETTERING CANC CTR,CELLULAR BIOCHEM & BIOPHYS PROGRAM,NEW YORK,NY 10021
Pavletich, NP
[J].
SCIENCE,
1996,
274
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[6]
THE P53 TUMOR SUPPRESSOR GENE
LEVINE, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Biology, Lewis Thomas Laboratory, Princeton University, Princeton
LEVINE, AJ
MOMAND, J
论文数:
0
引用数:
0
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