Structure and design of potent and selective cathepsin K inhibitors

被引：100

作者：

Yamashita, DS

Smith, WW

Zhao, BG

Janson, CA

Tomaszek, TA

Bossard, MJ

Levy, MA

Oh, HJ

Carr, TJ

Thompson, SK

Ijames, CF

Carr, SA

McQueney, M

DAlessio, KJ

Amegadzie, BY

Hanning, CR

AbdelMeguid, S

DesJarlais, RL

Gleason, JG

Veber, DF

机构：

[1] SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406

[2] SMITHKLINE BEECHAM PHARMACEUT,DEPT MACROMOL SCI,KING OF PRUSSIA,PA 19406

[3] SMITHKLINE BEECHAM PHARMACEUT,DEPT MOL RECOGNIT,KING OF PRUSSIA,PA 19406

[4] SMITHKLINE BEECHAM PHARMACEUT,DEPT PHYS & STRUCT CHEM,KING OF PRUSSIA,PA 19406

[5] SMITHKLINE BEECHAM PHARMACEUT,DEPT PROT BIOCHEM,KING OF PRUSSIA,PA 19406

[6] SMITHKLINE BEECHAM PHARMACEUT,DEPT GENE EXPRESS SCI,KING OF PRUSSIA,PA 19406

来源：

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY | 1997年 / 119卷 / 46期

关键词：

D O I：

10.1021/ja972204u

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

[No abstract available]

引用

页码：11351 / 11352

页数：2

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