Synthesis and biological activity of α-aminoboronic acids, amine-carboxyboranes and their derivatives

被引：65

作者：

Dembitsky, VM ^{[1
]}

Srebnik, M ^{[1
]}

机构：

[1] Hebrew Univ Jerusalem, Sch Pharm, Dept Med Chem & Nat Prod, IL-91120 Jerusalem, Israel

来源：

TETRAHEDRON | 2003年 / 59卷 / 05期

关键词：

alpha-aminoboronic acids; synthesis; serine proteases; amino-carboxyboranes inhibitors; boronic acids;

D O I：

10.1016/S0040-4020(02)01618-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[No abstract available]

引用

页码：579 / 593

页数：15

共 119 条

[51] NITRIC-OXIDE - A NEW PARADIGM FOR 2ND-MESSENGERS [J].

KERWIN, JF ;

LANCASTER, JR ;

FELDMAN, PL .

JOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (22) :4343-4362

[52]

KETTNER C, 1990, J BIOL CHEM, V265, P18289

[53] ACYLAMINO BORONIC ACIDS AND DIFLUOROBORANE ANALOGS OF AMINO-ACIDS - POTENT INHIBITORS OF CHYMOTRYPSIN AND ELASTASE [J].

KINDER, DH ;

KATZENELLENBOGEN, JA .

JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (12) :1917-1925

[54]

KNABB RM, 1992, THROMB HAEMOSTASIS, V67, P56

[55] SERINE PROTEASES - STRUCTURE AND MECHANISM OF CATALYSIS [J].

KRAUT, J .

ANNUAL REVIEW OF BIOCHEMISTRY, 1977, 46 :331-358

[56] PREDICTION OF NEW SERINE PROTEINASE-INHIBITORS [J].

KURINOV, IV ;

HARRISON, RW .

NATURE STRUCTURAL BIOLOGY, 1994, 1 (10) :735-743

[57] Hepatitis C virus NS3/4A protease [J].

Kwong, AD .

CURRENT OPINION IN INFECTIOUS DISEASES, 1997, 10 (06) :485-490

[58] Synthesis of boronic acid analogs of L-arginine as alternate substrates or inhibitors of nitric oxide synthase [J].

Lebarbier, C ;

Carreaux, F ;

Carboni, B ;

Boucher, JL .

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1998, 8 (18) :2573-2576

[59]

Lebarbier C, 1996, SYNTHESIS-STUTTGART, P1371

[60] AMINOMETHANEBORONIC ACIDS - SYNTHESIS AND INHIBITION OF A BORON ANALOG OF ESTERASE SUBSTRATES [J].

LINDQUIST, RN ;

NGUYEN, AC .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1977, 99 (19) :6435-6437

← 1 2 3 4 5 6 7 8 9 10 →