Studies on uracils:: an efficient method for the synthesis of novel 1-allyl-6-(1′,2′,3′-triazolyl) analogues of HEPT

被引：30

作者：

Bhuyan, PJ ^{[1
]}

Borah, HN ^{[1
]}

Sandhu, JS ^{[1
]}

机构：

[1] Reg Res Lab, Jorhat 785006, Assam, India

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 1999年 / 21期

关键词：

D O I：

10.1039/a906222j

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient synthetic method for preparing novel 1-allyl-6-(1',2',3'-triazolyl) analogues of HEPT, an anti-HIV reverse transcriptase inhibitor, is reported. The key step is based upon selective intermolecular cycloaddition of azide to acetylenes.

引用

页码：3083 / 3084

页数：2

共 24 条

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