Solution phase combinatorial synthesis of arylpiperazines

被引：38

作者：

Neuville, L ^{[1
]}

Zhu, JP ^{[1
]}

机构：

[1] CNRS,INST CHIM SUBST NAT,F-91198 GIF SUR YVETTE,FRANCE

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 23期

关键词：

D O I：

10.1016/S0040-4039(97)00831-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A solution phase combinatorial synthesis of aryl piperazines 1 and 2 is described based on the SNAr reaction and Schotten-Baumann acylation. The use of excess reagent is allowed and pure arylpiperazines 1 and 2 were obtained by simple acid/base washing. (C) 1997 Published by Elsevier Science Ltd.

引用

页码：4091 / 4094

页数：4

共 34 条

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