5-HT2C receptor modulation and the treatment of obesity

被引:36
作者
Bickerdike, MJ [1 ]
Vickers, SP [1 ]
Dourish, CT [1 ]
机构
[1] Cerebrus PLC, Wokingham RG41 5UA, England
关键词
D O I
10.1046/j.1463-1326.1999.00037.x
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
[No abstract available]
引用
收藏
页码:207 / 214
页数:8
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共 77 条
[51]  
Martin JR, 1998, J PHARMACOL EXP THER, V286, P913
[52]   Sibutramine - A review of its contribution to the management of obesity [J].
McNeely, W ;
Goa, KL .
DRUGS, 1998, 56 (06) :1093-1124
[53]  
MENNINI T, 1991, N-S ARCH PHARMACOL, V343, P483
[54]   5-HT1C RECEPTOR IS A PROMINENT SEROTONIN RECEPTOR SUBTYPE IN THE CENTRAL NERVOUS-SYSTEM [J].
MOLINEAUX, SM ;
JESSELL, TM ;
AXEL, R ;
JULIUS, D .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1989, 86 (17) :6793-6797
[55]   EVIDENCE THAT D-FENFLURAMINE ANOREXIA IS MEDIATED BY 5-HT1 RECEPTORS [J].
NEILL, JC ;
COOPER, SJ .
PSYCHOPHARMACOLOGY, 1989, 97 (02) :213-218
[56]   EFFECT OF CYPROHEPTADINE ON APPETITE AND WEIGHT GAIN IN ADULTS [J].
NOBLE, RE .
JOURNAL OF THE AMERICAN MEDICAL ASSOCIATION, 1969, 209 (13) :2054-&
[57]   Leptin-independent hyperphagia and type 2 diabetes in mice with a mutated serotonin 5-HT2C receptor gene [J].
Nonogaki, K ;
Strack, AM ;
Dallman, MF ;
Tecott, LH .
NATURE MEDICINE, 1998, 4 (10) :1152-1156
[58]   THE BINDING OF SEROTONERGIC LIGANDS TO THE PORCINE CHOROID-PLEXUS - CHARACTERIZATION OF A NEW TYPE OF SEROTONIN RECOGNITION SITE [J].
PAZOS, A ;
HOYER, D ;
PALACIOS, JM .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 106 (03) :539-546
[59]   Hypothalamic control of food intake in rats and cats - Prospective overview - Hypothalamus and the control of feeding: Fifteen decades of direct association [J].
Plata-Salaman, CR .
NUTRITION, 1998, 14 (01) :67-70
[60]  
ROSENZWEIGLIPSO.S, 1997, SOC NEUROSCI, V23