The first preparation of α-functionalized benzylamine

被引：15

作者：

Cho, SD

Kim, HJ

Ahn, CJ

Falck, JR ^{[1
]}

Shin, DS

机构：

[1] Changwon Natl Univ, Dept Chem, Changwon 641773, South Korea

[2] Univ Texas, SW Med Ctr, Dept Biochem, Dallas, TX 75235 USA

[3] Univ Texas, SW Med Ctr, Dept Pharmacol, Dallas, TX 75235 USA

来源：

TETRAHEDRON LETTERS | 1999年 / 40卷 / 47期

关键词：

D O I：

10.1016/S0040-4039(99)01713-X

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

We have investigated the alpha-acetoxylation of benzylamine derivatives 4 from substituted benzylphthalimide 3 using NBS/AcONa/AcOH in chlorobenzene at reflux. (C) 1999 Elsevier Science Ltd. All rights reserved.

引用

页码：8215 / 8217

页数：3

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