Solid-phase synthesis of branched thiohydantoin benzimidazolinethiones and branched thiohydantoin tetrahydroquinoxalinediones

被引：31

作者：

Nefzi, A ^{[1
]}

Giulianotti, MA ^{[1
]}

Houghten, RA ^{[1
]}

机构：

[1] Torrey Pines Inst Mol Studies, San Diego, CA 92121 USA

来源：

TETRAHEDRON LETTERS | 2000年 / 41卷 / 14期

关键词：

benzimidazolinethiones; solid-phase synthesis; tetrahydroquinoxalinediones; thiohydantoin;

D O I：

10.1016/S0040-4039(00)00162-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient solid-phase synthesis method is described for branched thiohydantoin benzimidazolinethiones and branched thiohydantoin tetrahydroquinoxalinediones using 4-fluoro-3-nitrobenzoic acid. (C) 2000 Elsevier Science Ltd. All rights reserved.

引用

页码：2283 / 2287

页数：5

共 22 条

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