French/European academic compound library initiative

被引：26

作者：

Hibert, Marcel F. ^{[1
]}

机构：

[1] Univ Strasbourg, UMR CNRS 7200, Fac Pharm, F-67401 Illkirch Graffenstaden, France

来源：

DRUG DISCOVERY TODAY | 2009年 / 14卷 / 15-16期

关键词：

INHIBITORS; LIGANDS;

D O I：

10.1016/j.drudis.2009.05.012

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：723 / 725

页数：3

共 11 条

[1] New biologically active linear triterpenes from the bark of three new-caledonian Cupaniopsis species [J].

Bousserouel, H ;

Litaudon, M ;

Morleo, B ;

Martin, MT ;

Thoison, O ;

Nosjean, O ;

Boutin, JA ;

Renard, P ;

Sévenet, T .

TETRAHEDRON, 2005, 61 (04) :845-851

[2] Use of a fluorescent polarization based high throughput assay to identify new Calmodulin ligands [J].

Dagher, Rania ;

Pigault, Claire ;

Bonnet, Dominique ;

Boeglin, Damien ;

Pourbaix, Christelle ;

Kilhoffer, Marie-Claude ;

Villa, Pascal ;

Wermuth, Camille G. ;

Hibert, Marcel ;

Haiech, Jacques .

BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR CELL RESEARCH, 2006, 1763 (11) :1250-1255

[3]

Hibert M., 2006, Patent, Patent No. [WO 2006003329 A1, 2006003329]

[4] Assessing the scaffold diversity of screening libraries [J].

Krier, M ;

Bret, G ;

Rognan, D .

JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2006, 46 (02) :512-524

[5] 3D-QSAR and docking studies of selective GSK-3,6 inhibitors.: Comparison with a thieno[2,3-b]pyrrolizinone derivative, a new potential lead for GSK-3,6 ligands [J].

Lescot, E ;

Bureau, R ;

Santos, JSD ;

Rochais, C ;

Lisowski, V ;

Lancelot, JC ;

Rault, S .

JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2005, 45 (03) :708-715

[6] A novel, conformation-specific allosteric inhibitor of the tachykinin NK2 receptor (NK2R) with functionally selective properties [J].

Maillet, Emeline L. ;

Pellegrini, Nadia ;

Valant, Celine ;

Bucher, Bernard ;

Hibert, Marcel ;

Bourguignon, Jean-Jacques ;

Galzi, Jean-Luc .

FASEB JOURNAL, 2007, 21 (09) :2124-2134

[7] Pharmacological inhibitors of glycogen synthase kinase 3 [J].

Meijer, L ;

Flajolet, M ;

Greengard, P .

TRENDS IN PHARMACOLOGICAL SCIENCES, 2004, 25 (09) :471-480

[8] Managing, profiling and analyzing a library of 2.6 million compounds gathered from 32 chemical providers [J].

Monge, Aurelien ;

Arrault, Alban ;

Marot, Christophe ;

Morin-Allory, Luc .

MOLECULAR DIVERSITY, 2006, 10 (03) :389-403

[9] Selective modification of alternative splicing by indole derivatives that target serine-arginine-rich protein splicing factors [J].

Soret, J ;

Bakkour, N ;

Maire, S ;

Durand, S ;

Zekri, L ;

Gabut, M ;

Fic, W ;

Divita, G ;

Rivalle, C ;

Dauzonne, D ;

Nguyen, CH ;

Jeanteur, P ;

Tazi, J .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2005, 102 (24) :8764-8769

[10] High-throughput screening in academia: The Harvard experience [J].

Stein, RL .

JOURNAL OF BIOMOLECULAR SCREENING, 2003, 8 (06) :615-619

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