Palladium-catalyzed functionalization of 5-and 7-azaindoles

被引：54

作者：

Chi, SM

Choi, JK

Yum, EK

Chi, DY

机构：

[1] Korea Res Inst Chem Technol, Bioorgan Sci Div, Yusung 305600, Taejeon, South Korea

[2] Inha Univ, Dept Chem, Inchon 402751, South Korea

来源：

TETRAHEDRON LETTERS | 2000年 / 41卷 / 06期

关键词：

D O I：

10.1016/S0040-4039(99)02190-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Palladium-catalyzed functionalization at the 2-position of various 5- and 7-azaindoles was performed by Suzuki, Heck, and Stille reactions. The 2-substituted azaindoles were obtained with 5% Pd(OAc)(2), LiCl, and KOAc in DMF at 110 degrees C with moderate to high yields. (C) 2000 Elsevier Science Ltd. All rights reserved.

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页码：919 / 922

页数：4

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