Biochemical and pharmacologic rationale for the development of a synthetic heparin pentasaccharide

被引:94
作者
Walenga, JM [1 ]
Jeske, WP [1 ]
Bara, L [1 ]
Samama, MM [1 ]
Fareed, J [1 ]
机构
[1] HOP HOTEL DIEU, DEPT BIOL HAEMATOL, PARIS, FRANCE
关键词
heparin; pentasaccharide; antithrombin; factor Xa; antithrombotic;
D O I
10.1016/S0049-3848(97)00042-X
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
[No abstract available]
引用
收藏
页码:1 / 36
页数:36
相关论文
共 140 条
[61]  
Jeske W., 1996, Blood, V88, p317A
[62]  
JESKE W, 1996, THESIS LOYOLA U CHIC
[63]   Initiation of the tissue factor pathway of coagulation in the presence of heparin: Control by antithrombin III and tissue factor pathway inhibitor [J].
Jesty, J ;
Lorenz, A ;
Rodriguez, J ;
Wun, TC .
BLOOD, 1996, 87 (06) :2301-2307
[64]  
JORDAN RE, 1980, J BIOL CHEM, V255, P81
[65]   INHIBITORY EFFECTS OF TFPI ON THROMBIN AND FACTOR XA GENERATION IN-VITRO - MODULATORY ACTION OF GLYCOSAMINOGLYCANS [J].
KAISER, B ;
HOPPENSTEADT, DA ;
JESKE, W ;
WUN, TC ;
FAREED, J .
THROMBOSIS RESEARCH, 1994, 75 (06) :609-616
[66]  
Kaiser B., 1996, Fibrinolysis, V10, P127
[67]  
KAISER B, 1993, THROMB HAEMOSTASIS, V69, P1111
[68]  
LABROUCHE S, 1992, THROMB HAEMOSTASIS, V68, P556
[69]   SEPARATION OF ACTIVE AND INACTIVE FORMS OF HEPARIN [J].
LAM, LH ;
SILBERT, JE ;
ROSENBERG, RD .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1976, 69 (02) :570-577
[70]   INTERACTION BETWEEN POLYSACCHARIDES AND OTHER MACROMOLECULES .27. MOLECULAR-WEIGHT-DEPENDENCE OF ANTI-COAGULANT ACTIVITY OF HEPARIN [J].
LAURENT, TC ;
TENGBLAD, A ;
THUNBERG, L ;
HOOK, M ;
LINDAHL, U .
BIOCHEMICAL JOURNAL, 1978, 175 (02) :691-701