Neat formic acid:: An excellent N-formylating agent for carbazoles, 3-alkylindoles, diphenylamine and moderately weak nucleophilic anilines

被引：19

作者：

Chakrabarty, M

Khasnobis, S

Harigaya, Y

Konda, Y

机构：

[1] Bose Inst, Dept Chem, Calcutta 700009, W Bengal, India

[2] Kitasato Univ, Sch Pharmaceut Sci, Minato Ku, Tokyo 108, Japan

来源：

SYNTHETIC COMMUNICATIONS | 2000年 / 30卷 / 02期

关键词：

D O I：

10.1080/00397910008087310

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Neat formic acid alone efficiently N-formylates carbazoles, 3-alkylindoles, diphenylamine and even moderately weak nucleophilic anilines to furnish the corresponding N-formyl derivatives in 72-87% yields.

引用

页码：187 / 200

页数：14

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