Synthesis of 3-methyl-substituted pyrazolotriazolopyrimidin-4-one and pyrazolothiazolopyrimidin-4-one derivatives

被引：12

作者：

Guccione, S ^{[1
]}

Scolaro, LM ^{[1
]}

Russo, F ^{[1
]}

机构：

[1] UNIV MESSINA,DIPARTIMENTO CHIM INORGAN ANAL & STRUTTURA MOLEC,SEZIONE MESSINA,I-98166 MESSINA,ITALY

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1996年 / 33卷 / 02期

关键词：

D O I：

10.1002/jhet.5570330239

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

As a part of a research on anti-inflammatory analgesic compounds 3-methyl substituted pyrazolotriazolopyrimidin-4-one and pyrazolothiazolopyrimidin-4-one derivatives were prepared by previously reported procedures. None of the compounds showed improved activity when compared with the previously reported unsubstituted analogs.

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页码：459 / 463

页数：5

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