N-acylation in combinatorial chemistry

被引：37

作者：

Katritzky, AR ^{[1
]}

Suzuki, K ^{[1
]}

Singh, SK ^{[1
]}

机构：

[1] Univ Florida, Dept Chem, Ctr Heterocycl Cpds, Gainesville, FL 32611 USA

来源：

ARKIVOC | 2004年

关键词：

N-acylation; N-acylating reagents; solid-phase; polymer-supported; combinatorial chemistry;

D O I：

10.3998/ark.5550190.0005.102

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Polymer-supported N-acylation utilizing carbodiimides with additives, direct coupling reagents ( phosphonium salts and uronium salts), N-acylazoles, and other reagents have been discussed.

引用

页码：12 / 35

页数：24

共 135 条

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