Syntheses of stereochemically diverse nine-membered ring-containing biaryls

被引：30

作者：

Krishnan, S ^{[1
]}

Schreiber, SL

机构：

[1] Harvard Univ, Howard Hughes Med Inst, Dept Chem & Chem Biol, Cambridge, MA 02138 USA

[2] Harvard Univ, Broad Inst, Cambridge, MA 02138 USA

[3] MIT, Cambridge, MA 02138 USA

来源：

ORGANIC LETTERS | 2004年 / 6卷 / 22期

关键词：

D O I：

10.1021/ol048273c

中图分类号：

O62 [有机化学];

学科分类号：

070303 [有机化学]; 081704 [应用化学];

摘要：

A library of nine-membered, biaryl-containing rings has been synthesized in parallel on polystyrene macrobeads. Dimeric medium rings were shown to be accessible via a regio- and stereoselective double cyclization.

引用

页码：4021 / 4024

页数：4

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