New synthesis of 3-substituted indazoles from 3-trimethylsilylindazole

被引：12

作者：

Hari, Y ^{[1
]}

Shoji, Y ^{[1
]}

Aoyama, T ^{[1
]}

机构：

[1] Nagoya City Univ, Grad Sch Pharmaceut Sci, Mizuho Ku, Nagoya, Aichi 4678603, Japan

来源：

SYNTHESIS-STUTTGART | 2004年 / 08期

关键词：

aryl aldehydes; Brook rearrangement; cesium fluoride; indazoles; silyl compounds;

D O I：

10.1055/s-2004-822531

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Reaction of aryl aldehydes with 3-trimethylsilylindazole in the presence of CsF easily gave the corresponding 3-(arylhydroxymethyl)indazoles in good to moderate yields.

引用

页码：1183 / 1186

页数：4

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