Polyaniline supported cobalt catalysed one pot stereoselective synthesis of the structural analogues of aminopeptidase inhibitor Bestatin

被引：23

作者：

De, A ^{[1
]}

Basak, P ^{[1
]}

Iqbal, J ^{[1
]}

机构：

[1] INDIAN INST TECHNOL, DEPT CHEM, KANPUR 208016, UTTAR PRADESH, INDIA

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 48期

关键词：

D O I：

10.1016/S0040-4039(97)10172-1

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A one pot stereoselective conversion of cinnamoyl amide of L-leucine methyl ester to the corresponding structural analogues of bestatin was achieved by employing polyaniline supported cobalt(II) salen catalysed epoxidation followed by its opening with anilines at ambient conditions. (C) 1997 Elsevier Science Ltd.

引用

页码：8383 / 8386

页数：4

共 14 条

[1] INHIBITION OF ENKEPHALIN-DEGRADING AMINOPEPTIDASE ACTIVITY BY CERTAIN PEPTIDES
BARCLAY, RK
PHILLIPPS, MA
[J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1980, 96 (04) : 1732 - 1738
[2] A cobalt catalyzed protocol for the synthesis of substituted beta-phenyl isoserine derivatives
Bhatia, B
Jain, S
De, A
Bagchi, I
Iqbal, J
[J]. TETRAHEDRON LETTERS, 1996, 37 (40) : 7311 - 7314
[3] Polyaniline supported cobalt(II) catalyst: Oxidation of alkenes with molecular oxygen
Das, BC
Iqbal, J
[J]. TETRAHEDRON LETTERS, 1997, 38 (07) : 1235 - 1238
[4] Polyaniline supported cobalt(II)-salen catalyst: One pot synthesis of beta-phenylisoserine derivatives from cinnamoyl amide
Das, BC
Iqbal, J
[J]. TETRAHEDRON LETTERS, 1997, 38 (16) : 2903 - 2906
[5] EFFECT OF BESTATIN ON INVITRO RESPONSES OF MURINE LYMPHOCYTES TO T-CELL STIMULI
DUNLAP, BE
DUNLAP, SA
RICH, DH
[J]. SCANDINAVIAN JOURNAL OF IMMUNOLOGY, 1984, 20 (03) : 237 - 245
[6] ADDITION OF AMINO ESTERS TO THIIRANIUM ION INTERMEDIATES - A NOVEL-APPROACH TO THE SYNTHESIS OF NEW POTENTIAL AMINOPEPTIDASE INHIBITORS
GILL, DM
PEGG, NA
RAYNER, CM
[J]. TETRAHEDRON LETTERS, 1995, 36 (45) : 8327 - 8330
[7] IDENTIFICATION AND PROPERTIES OF THE CELL-MEMBRANE BOUND LEUCINE AMINOPEPTIDASE INTERACTING WITH THE POTENTIAL IMMUNOSTIMULANT AND CHEMOTHERAPEUTIC AGENT BESTATIN
LEYHAUSEN, G
SCHUSTER, DK
VAITH, P
ZAHN, RK
UMEZAWA, H
FALKE, D
MULLER, WEG
[J]. BIOCHEMICAL PHARMACOLOGY, 1983, 32 (06) : 1051 - 1057
[8] SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF BESTATIN ANALOGS, INHIBITORS OF AMINOPEPTIDASE-B
NISHIZAWA, R
SAINO, T
TAKITA, T
SUDA, H
AOYAGI, T
UMEZAWA, H
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1977, 20 (04) : 510 - 515
[9] A STEREOSPECIFIC SYNTHESIS OF (-)-BESTATIN FROM L-MALIC ACID
NORMAN, BH
MORRIS, ML
[J]. TETRAHEDRON LETTERS, 1992, 33 (45) : 6803 - 6806
[10] PUNNIYAMURTHY T, 1997, TETRAHEDRON LETT, V38, P4466

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