A new approach to the solid-phase Suzuki coupling reaction.

被引：77

作者：

Piettre, SR

Baltzer, S

机构：

[1] Marion Merrell Research Institute, Strasbourg Research Center, 67080 Strasbourg

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 07期

关键词：

D O I：

10.1016/S0040-4039(97)00063-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Treatment of polymer-bound aryl halides with pinacol ester of diboron under palladium (0) catalysis gave the corresponding polymer-bound boronates. The Suzuki coupling reaction was then carried out using a variety of aryl halides. Cleavage from the solid support delivered the expected products in usually good yields and high purity. (C) 1997, Published by Elsevier Science Ltd.

引用

页码：1197 / 1200

页数：4

共 23 条

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