Synthesis and reactivity of azaindoles: Applications in the preparation of bioactive molecules

被引：16

作者：

Le Hyaric, M ^{[1
]}

de Almeida, MV ^{[1
]}

de Souza, MVN ^{[1
]}

机构：

[1] Univ Fed Juiz de Fora, Inst Ciencias Exatas, Dept Quim, BR-36038330 Juiz de Fora, MG, Brazil

来源：

QUIMICA NOVA | 2002年 / 25卷 / 6B期

关键词：

azaindole; synthetic methods; biological activity;

D O I：

10.1590/S0100-40422002000700017

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Synthetic methods used for the preparation of azaindoles are described in this article. Applications in the preparation of bioactive molecules are given: synthesis of substituted 6-azaindoles as benzodiazepines receptor ligands, substituted 7-azaindoles as dopamine D-4 ligands and preparation of an olivacine analogue.

引用

页码：1165 / 1171

页数：7

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