Studies on the selective intramolecular biaryl coupling reaction of 2-triflyloxy-6-halobenzanilides using a palladium reagent

被引：7

作者：

Harayama, T ^{[1
]}

Toko, H ^{[1
]}

Kubota, K ^{[1
]}

Nishioka, H ^{[1
]}

Abe, H ^{[1
]}

Takeuchi, Y ^{[1
]}

机构：

[1] Okayama Univ, Fac Pharmaceut Sci, Okayama 7008530, Japan

来源：

HETEROCYCLES | 2002年 / 58卷

关键词：

D O I：

10.3987/COM-01-S(M)5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The aryl-aryl coupling reaction of 2-triflyloxy-6-halobenzanilides using a palladium reagent under several reaction conditions was examined. The 6-iodo compound gave triflyloxyphenanthridone selectively in excellent yield under the conditions for the ordinary Heck reaction.

引用

页码：175 / 181

页数：7

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