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Induction of P-glycoprotein expression by HIV protease inhibitors in cell culture
被引:77
作者
:
Perloff, MD
论文数:
0
引用数:
0
h-index:
0
机构:
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
Perloff, MD
[
1
]
von Moltke, LL
论文数:
0
引用数:
0
h-index:
0
机构:
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
von Moltke, LL
Fahey, JM
论文数:
0
引用数:
0
h-index:
0
机构:
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
Fahey, JM
Daily, JP
论文数:
0
引用数:
0
h-index:
0
机构:
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
Daily, JP
Greenblatt, DJ
论文数:
0
引用数:
0
h-index:
0
机构:
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
Greenblatt, DJ
机构
:
[1]
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
[2]
New England Med Ctr, Div Clin Pharmacol, Boston, MA 02111 USA
[3]
Harvard Univ, Sch Med, Dept Med, Boston, MA 02115 USA
[4]
Brigham & Womens Hosp, Boston, MA 02115 USA
来源
:
AIDS
|
2000年
/ 14卷
/ 09期
关键词
:
D O I
:
10.1097/00002030-200006160-00034
中图分类号
:
R392 [医学免疫学];
Q939.91 [免疫学];
学科分类号
:
100102 ;
摘要
:
引用
收藏
页码:1287 / 1289
页数:3
相关论文
共 15 条
[1]
P-glycoprotein and multidrug resistance
[J].
Gottesman, MM
论文数:
0
引用数:
0
h-index:
0
机构:
NCI,NIH,DIV BASIC SCI,MOL BIOL LAB,BETHESDA,MD 20892
NCI,NIH,DIV BASIC SCI,MOL BIOL LAB,BETHESDA,MD 20892
Gottesman, MM
;
Pastan, I
论文数:
0
引用数:
0
h-index:
0
机构:
NCI,NIH,DIV BASIC SCI,MOL BIOL LAB,BETHESDA,MD 20892
NCI,NIH,DIV BASIC SCI,MOL BIOL LAB,BETHESDA,MD 20892
Pastan, I
;
Ambudkar, SV
论文数:
0
引用数:
0
h-index:
0
机构:
NCI,NIH,DIV BASIC SCI,MOL BIOL LAB,BETHESDA,MD 20892
NCI,NIH,DIV BASIC SCI,MOL BIOL LAB,BETHESDA,MD 20892
Ambudkar, SV
.
CURRENT OPINION IN GENETICS & DEVELOPMENT,
1996,
6
(05)
:610
-617
[2]
P-GLYCOPROTEIN EXPRESSION AND REGULATION - AGE-RELATED-CHANGES AND POTENTIAL EFFECTS ON DRUG-THERAPY
[J].
GUPTA, S
论文数:
0
引用数:
0
h-index:
0
机构:
Division of Basic and Clinical Immunology, University of California, Irvine, California
GUPTA, S
.
DRUGS & AGING,
1995,
7
(01)
:19
-29
[3]
Interactions of HIV protease inhibitors with ATP-dependent drug export proteins
[J].
Gutmann, H
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS, Lab Pharmacol & Chem, NIH, Res Triangle Pk, NC 27709 USA
Gutmann, H
;
Fricker, G
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS, Lab Pharmacol & Chem, NIH, Res Triangle Pk, NC 27709 USA
Fricker, G
;
Drewe, J
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS, Lab Pharmacol & Chem, NIH, Res Triangle Pk, NC 27709 USA
Drewe, J
;
Toeroek, M
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS, Lab Pharmacol & Chem, NIH, Res Triangle Pk, NC 27709 USA
Toeroek, M
;
Miller, DS
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS, Lab Pharmacol & Chem, NIH, Res Triangle Pk, NC 27709 USA
Miller, DS
.
MOLECULAR PHARMACOLOGY,
1999,
56
(02)
:383
-389
[4]
HERZOG CE, 1993, J BIOL CHEM, V268, P2946
[5]
The drug transporter P-glycoprotein limits oral absorption and brain entry of HIV-1 protease inhibitors
[J].
Kim, RB
论文数:
0
引用数:
0
h-index:
0
机构:
Vanderbilt Univ, Sch Med, Div Clin Pharmacol, Dept Med, Nashville, TN 37232 USA
Kim, RB
;
Fromm, MF
论文数:
0
引用数:
0
h-index:
0
机构:
Vanderbilt Univ, Sch Med, Div Clin Pharmacol, Dept Med, Nashville, TN 37232 USA
Fromm, MF
;
Wandel, C
论文数:
0
引用数:
0
h-index:
0
机构:
Vanderbilt Univ, Sch Med, Div Clin Pharmacol, Dept Med, Nashville, TN 37232 USA
Wandel, C
;
Leake, B
论文数:
0
引用数:
0
h-index:
0
机构:
Vanderbilt Univ, Sch Med, Div Clin Pharmacol, Dept Med, Nashville, TN 37232 USA
Leake, B
;
Wood, AJJ
论文数:
0
引用数:
0
h-index:
0
机构:
Vanderbilt Univ, Sch Med, Div Clin Pharmacol, Dept Med, Nashville, TN 37232 USA
Wood, AJJ
;
Roden, DM
论文数:
0
引用数:
0
h-index:
0
机构:
Vanderbilt Univ, Sch Med, Div Clin Pharmacol, Dept Med, Nashville, TN 37232 USA
Roden, DM
;
Wilkinson, GR
论文数:
0
引用数:
0
h-index:
0
机构:
Vanderbilt Univ, Sch Med, Div Clin Pharmacol, Dept Med, Nashville, TN 37232 USA
Wilkinson, GR
.
JOURNAL OF CLINICAL INVESTIGATION,
1998,
101
(02)
:289
-294
[6]
HIV-1 protease inhibitors and the MDR1 multidrug transporter
[J].
Lee, CGL
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Lee, CGL
;
Gottesman, MM
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Gottesman, MM
.
JOURNAL OF CLINICAL INVESTIGATION,
1998,
101
(02)
:287
-288
[7]
HIV-1 protease inhibitors are substrates for the MDR1 multidrug transporter
[J].
Lee, CGL
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Lee, CGL
;
Gottesman, MM
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Gottesman, MM
;
Cardarelli, CO
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Cardarelli, CO
;
Ramachandra, M
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Ramachandra, M
;
Jeang, KT
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Jeang, KT
;
Ambudkar, SV
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Ambudkar, SV
;
Pastan, I
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Pastan, I
;
Dey, S
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Dey, S
.
BIOCHEMISTRY,
1998,
37
(11)
:3594
-3601
[8]
Unchanged cytochrome P450 3A (CYP3A) expression and metabolism of midazolam, triazolam, and dexamethasone in mdr(-/-) mouse liver microsomes
[J].
Perloff, MD
论文数:
0
引用数:
0
h-index:
0
机构:
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
Perloff, MD
;
von Moltke, LL
论文数:
0
引用数:
0
h-index:
0
机构:
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
von Moltke, LL
;
Cotreau, MM
论文数:
0
引用数:
0
h-index:
0
机构:
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
Cotreau, MM
;
Greenblatt, DJ
论文数:
0
引用数:
0
h-index:
0
机构:
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
Greenblatt, DJ
.
BIOCHEMICAL PHARMACOLOGY,
1999,
57
(11)
:1227
-1232
[9]
MULTIDRUG TRANSPORTER P-GLYCOPROTEIN-170 AS A DIFFERENTIATION ANTIGEN ON NORMAL HUMAN-LYMPHOCYTES AND THYMOCYTES - MODULATION WITH DIFFERENTIATION STAGE AND DURING AGING
[J].
PILARSKI, LM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ALBERTA,DEPT MED,EDMONTON,AB TG6 1Z2,CANADA
PILARSKI, LM
;
PAINE, D
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ALBERTA,DEPT MED,EDMONTON,AB TG6 1Z2,CANADA
PAINE, D
;
MCELHANEY, JE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ALBERTA,DEPT MED,EDMONTON,AB TG6 1Z2,CANADA
MCELHANEY, JE
;
CASS, CE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ALBERTA,DEPT MED,EDMONTON,AB TG6 1Z2,CANADA
CASS, CE
;
BELCH, AR
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ALBERTA,DEPT MED,EDMONTON,AB TG6 1Z2,CANADA
BELCH, AR
.
AMERICAN JOURNAL OF HEMATOLOGY,
1995,
49
(04)
:323
-335
[10]
Modulation of P-glycoprotein function in human lymphocytes and Caco-2 cell monolayers by HIV-1 protease inhibitors
[J].
Profit, L
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Liverpool, Dept Pharmacol & Therapeut, Liverpool L69 3GE, Merseyside, England
Univ Liverpool, Dept Pharmacol & Therapeut, Liverpool L69 3GE, Merseyside, England
Profit, L
;
Eagling, VA
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Liverpool, Dept Pharmacol & Therapeut, Liverpool L69 3GE, Merseyside, England
Univ Liverpool, Dept Pharmacol & Therapeut, Liverpool L69 3GE, Merseyside, England
Eagling, VA
;
Back, DJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Liverpool, Dept Pharmacol & Therapeut, Liverpool L69 3GE, Merseyside, England
Univ Liverpool, Dept Pharmacol & Therapeut, Liverpool L69 3GE, Merseyside, England
Back, DJ
.
AIDS,
1999,
13
(13)
:1623
-1627
←
1
2
→
共 15 条
[1]
P-glycoprotein and multidrug resistance
[J].
Gottesman, MM
论文数:
0
引用数:
0
h-index:
0
机构:
NCI,NIH,DIV BASIC SCI,MOL BIOL LAB,BETHESDA,MD 20892
NCI,NIH,DIV BASIC SCI,MOL BIOL LAB,BETHESDA,MD 20892
Gottesman, MM
;
Pastan, I
论文数:
0
引用数:
0
h-index:
0
机构:
NCI,NIH,DIV BASIC SCI,MOL BIOL LAB,BETHESDA,MD 20892
NCI,NIH,DIV BASIC SCI,MOL BIOL LAB,BETHESDA,MD 20892
Pastan, I
;
Ambudkar, SV
论文数:
0
引用数:
0
h-index:
0
机构:
NCI,NIH,DIV BASIC SCI,MOL BIOL LAB,BETHESDA,MD 20892
NCI,NIH,DIV BASIC SCI,MOL BIOL LAB,BETHESDA,MD 20892
Ambudkar, SV
.
CURRENT OPINION IN GENETICS & DEVELOPMENT,
1996,
6
(05)
:610
-617
[2]
P-GLYCOPROTEIN EXPRESSION AND REGULATION - AGE-RELATED-CHANGES AND POTENTIAL EFFECTS ON DRUG-THERAPY
[J].
GUPTA, S
论文数:
0
引用数:
0
h-index:
0
机构:
Division of Basic and Clinical Immunology, University of California, Irvine, California
GUPTA, S
.
DRUGS & AGING,
1995,
7
(01)
:19
-29
[3]
Interactions of HIV protease inhibitors with ATP-dependent drug export proteins
[J].
Gutmann, H
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS, Lab Pharmacol & Chem, NIH, Res Triangle Pk, NC 27709 USA
Gutmann, H
;
Fricker, G
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS, Lab Pharmacol & Chem, NIH, Res Triangle Pk, NC 27709 USA
Fricker, G
;
Drewe, J
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS, Lab Pharmacol & Chem, NIH, Res Triangle Pk, NC 27709 USA
Drewe, J
;
Toeroek, M
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS, Lab Pharmacol & Chem, NIH, Res Triangle Pk, NC 27709 USA
Toeroek, M
;
Miller, DS
论文数:
0
引用数:
0
h-index:
0
机构:
NIEHS, Lab Pharmacol & Chem, NIH, Res Triangle Pk, NC 27709 USA
Miller, DS
.
MOLECULAR PHARMACOLOGY,
1999,
56
(02)
:383
-389
[4]
HERZOG CE, 1993, J BIOL CHEM, V268, P2946
[5]
The drug transporter P-glycoprotein limits oral absorption and brain entry of HIV-1 protease inhibitors
[J].
Kim, RB
论文数:
0
引用数:
0
h-index:
0
机构:
Vanderbilt Univ, Sch Med, Div Clin Pharmacol, Dept Med, Nashville, TN 37232 USA
Kim, RB
;
Fromm, MF
论文数:
0
引用数:
0
h-index:
0
机构:
Vanderbilt Univ, Sch Med, Div Clin Pharmacol, Dept Med, Nashville, TN 37232 USA
Fromm, MF
;
Wandel, C
论文数:
0
引用数:
0
h-index:
0
机构:
Vanderbilt Univ, Sch Med, Div Clin Pharmacol, Dept Med, Nashville, TN 37232 USA
Wandel, C
;
Leake, B
论文数:
0
引用数:
0
h-index:
0
机构:
Vanderbilt Univ, Sch Med, Div Clin Pharmacol, Dept Med, Nashville, TN 37232 USA
Leake, B
;
Wood, AJJ
论文数:
0
引用数:
0
h-index:
0
机构:
Vanderbilt Univ, Sch Med, Div Clin Pharmacol, Dept Med, Nashville, TN 37232 USA
Wood, AJJ
;
Roden, DM
论文数:
0
引用数:
0
h-index:
0
机构:
Vanderbilt Univ, Sch Med, Div Clin Pharmacol, Dept Med, Nashville, TN 37232 USA
Roden, DM
;
Wilkinson, GR
论文数:
0
引用数:
0
h-index:
0
机构:
Vanderbilt Univ, Sch Med, Div Clin Pharmacol, Dept Med, Nashville, TN 37232 USA
Wilkinson, GR
.
JOURNAL OF CLINICAL INVESTIGATION,
1998,
101
(02)
:289
-294
[6]
HIV-1 protease inhibitors and the MDR1 multidrug transporter
[J].
Lee, CGL
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Lee, CGL
;
Gottesman, MM
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Gottesman, MM
.
JOURNAL OF CLINICAL INVESTIGATION,
1998,
101
(02)
:287
-288
[7]
HIV-1 protease inhibitors are substrates for the MDR1 multidrug transporter
[J].
Lee, CGL
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Lee, CGL
;
Gottesman, MM
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Gottesman, MM
;
Cardarelli, CO
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Cardarelli, CO
;
Ramachandra, M
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Ramachandra, M
;
Jeang, KT
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Jeang, KT
;
Ambudkar, SV
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Ambudkar, SV
;
Pastan, I
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Pastan, I
;
Dey, S
论文数:
0
引用数:
0
h-index:
0
机构:
NCI, Cell Biol Lab, NIH, Bethesda, MD 20892 USA
Dey, S
.
BIOCHEMISTRY,
1998,
37
(11)
:3594
-3601
[8]
Unchanged cytochrome P450 3A (CYP3A) expression and metabolism of midazolam, triazolam, and dexamethasone in mdr(-/-) mouse liver microsomes
[J].
Perloff, MD
论文数:
0
引用数:
0
h-index:
0
机构:
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
Perloff, MD
;
von Moltke, LL
论文数:
0
引用数:
0
h-index:
0
机构:
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
von Moltke, LL
;
Cotreau, MM
论文数:
0
引用数:
0
h-index:
0
机构:
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
Cotreau, MM
;
Greenblatt, DJ
论文数:
0
引用数:
0
h-index:
0
机构:
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
Tufts Univ, Sch Med, Dept Pharmacol & Expt Therapeut, Boston, MA 02111 USA
Greenblatt, DJ
.
BIOCHEMICAL PHARMACOLOGY,
1999,
57
(11)
:1227
-1232
[9]
MULTIDRUG TRANSPORTER P-GLYCOPROTEIN-170 AS A DIFFERENTIATION ANTIGEN ON NORMAL HUMAN-LYMPHOCYTES AND THYMOCYTES - MODULATION WITH DIFFERENTIATION STAGE AND DURING AGING
[J].
PILARSKI, LM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ALBERTA,DEPT MED,EDMONTON,AB TG6 1Z2,CANADA
PILARSKI, LM
;
PAINE, D
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ALBERTA,DEPT MED,EDMONTON,AB TG6 1Z2,CANADA
PAINE, D
;
MCELHANEY, JE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ALBERTA,DEPT MED,EDMONTON,AB TG6 1Z2,CANADA
MCELHANEY, JE
;
CASS, CE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ALBERTA,DEPT MED,EDMONTON,AB TG6 1Z2,CANADA
CASS, CE
;
BELCH, AR
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ALBERTA,DEPT MED,EDMONTON,AB TG6 1Z2,CANADA
BELCH, AR
.
AMERICAN JOURNAL OF HEMATOLOGY,
1995,
49
(04)
:323
-335
[10]
Modulation of P-glycoprotein function in human lymphocytes and Caco-2 cell monolayers by HIV-1 protease inhibitors
[J].
Profit, L
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Liverpool, Dept Pharmacol & Therapeut, Liverpool L69 3GE, Merseyside, England
Univ Liverpool, Dept Pharmacol & Therapeut, Liverpool L69 3GE, Merseyside, England
Profit, L
;
Eagling, VA
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Liverpool, Dept Pharmacol & Therapeut, Liverpool L69 3GE, Merseyside, England
Univ Liverpool, Dept Pharmacol & Therapeut, Liverpool L69 3GE, Merseyside, England
Eagling, VA
;
Back, DJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Liverpool, Dept Pharmacol & Therapeut, Liverpool L69 3GE, Merseyside, England
Univ Liverpool, Dept Pharmacol & Therapeut, Liverpool L69 3GE, Merseyside, England
Back, DJ
.
AIDS,
1999,
13
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:1623
-1627
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