Enhanced release of itraconazole from ordered mesoporous SBA-15 silica materials

被引:200
作者
Mellaerts, Randy
Aerts, Caroline A.
Van Humbeeck, Jan
Augustijns, Patrick
Van den Mooter, Guy
Martens, Johan A.
机构
[1] Catholic Univ Leuven, Ctr Surface Chem & Catalysis, BE-3001 Heverlee, Belgium
[2] Catholic Univ Leuven, Dept Met & Mat Engn, BE-3001 Heverlee, Belgium
[3] Catholic Univ Louvain, Lab Pharmacotechnol & Biopharm, BE-3000 Louvain, Belgium
关键词
D O I
10.1039/b616746b
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
This in vitro study reports on the enhanced release of the hydrophobic drug itraconazole from the ordered mesoporous SBA-15 silica material and on the existence of a critical mesopore diameter for enhancing release.
引用
收藏
页码:1375 / 1377
页数:3
相关论文
共 17 条
[1]   Influences of material characteristics on ibuprofen drug loading and release profiles from ordered micro- and mesoporous silica matrices [J].
Andersson, J ;
Rosenholm, J ;
Areva, S ;
Lindén, M .
CHEMISTRY OF MATERIALS, 2004, 16 (21) :4160-4167
[2]   A NEW FAMILY OF MESOPOROUS MOLECULAR-SIEVES PREPARED WITH LIQUID-CRYSTAL TEMPLATES [J].
BECK, JS ;
VARTULI, JC ;
ROTH, WJ ;
LEONOWICZ, ME ;
KRESGE, CT ;
SCHMITT, KD ;
CHU, CTW ;
OLSON, DH ;
SHEPPARD, EW ;
MCCULLEN, SB ;
HIGGINS, JB ;
SCHLENKER, JL .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1992, 114 (27) :10834-10843
[3]   Mesoporous silica material TUD-1 as a drug delivery system [J].
Heikkila, T. ;
Salonen, J. ;
Tuura, J. ;
Hamdy, M. S. ;
Mul, G. ;
Kumar, N. ;
Salmi, T. ;
Murzin, D. Yu ;
Laitinen, L. ;
Kaukonen, A. M. ;
Hirvonen, J. ;
Lehto, V. -P. .
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2007, 331 (01) :133-138
[4]   Influence of pore size of MCM-41 matrices on drug delivery rate [J].
Horcajada, P ;
Rámila, A ;
Pérez-Pariente, J ;
Vallet-Regí, M .
MICROPOROUS AND MESOPOROUS MATERIALS, 2004, 68 (1-3) :105-109
[5]  
Kortesuo P, 1999, J BIOMED MATER RES, V44, P162, DOI 10.1002/(SICI)1097-4636(199902)44:2<162::AID-JBM6>3.0.CO
[6]  
2-P
[7]   Improving drug solubility for oral delivery using solid dispersions [J].
Leuner, C ;
Dressman, J .
EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS, 2000, 50 (01) :47-60
[8]   Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings [J].
Lipinski, CA ;
Lombardo, F ;
Dominy, BW ;
Feeney, PJ .
ADVANCED DRUG DELIVERY REVIEWS, 1997, 23 (1-3) :3-25
[9]   Pharmaceutical applications of cyclodextrins .1. Drug solubilization and stabilization [J].
Loftsson, T ;
Brewster, ME .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1996, 85 (10) :1017-1025
[10]   Formulation of self-emulsifying drug delivery systems [J].
Pouton, CW .
ADVANCED DRUG DELIVERY REVIEWS, 1997, 25 (01) :47-58