Rapid analogue syntheses of heteroaromatic compounds

被引：67

作者：

Collins, I ^{[1
]}

机构：

[1] Merck Sharp & Dohme Res Labs, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 2000年 / 17期

关键词：

D O I：

10.1039/a904715h

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Recent advances in the practical and rapid synthesis of multiply substituted aromatic heterocycles were reviewed. Focus was on bond formation to ring atoms as opposed to the modification of side-chains. Work on the solution-phase synthesis of 5- and 6-membered heteroaromatic compounds and their fused derivatives were discussed.

引用

页码：2845 / 2861

页数：17

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