Rapid analogue syntheses of heteroaromatic compounds

被引:67
作者
Collins, I [1 ]
机构
[1] Merck Sharp & Dohme Res Labs, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England
来源
JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 2000年 / 17期
关键词
D O I
10.1039/a904715h
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Recent advances in the practical and rapid synthesis of multiply substituted aromatic heterocycles were reviewed. Focus was on bond formation to ring atoms as opposed to the modification of side-chains. Work on the solution-phase synthesis of 5- and 6-membered heteroaromatic compounds and their fused derivatives were discussed.
引用
收藏
页码:2845 / 2861
页数:17
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