Synthesis of new melatonin analogues from dimers of azaindole and indole by use of Suzuki homocoupling

被引：15

作者：

Guillard, J ^{[1
]}

Larraya, C ^{[1
]}

Viaud-Massuard, MC ^{[1
]}

机构：

[1] Univ Tours, UFR Sci Pharmaceut, GRCHT Lab Chim ORgan, EA 3247, F-37200 Tours, France

来源：

HETEROCYCLES | 2003年 / 60卷 / 04期

关键词：

D O I：

10.3987/COM-02-9695

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

N-{2-[3'-(2-Acetylaminoethyl)-1H,1'H-[5,5']biindol-3-yl]- and N-{2-[1'-(2-acetylaminoethyl)-1'H-[5,5']biindol-1-yl]ethyl}acetamide (2,3) and their analogues in 7-azaindole series (4,5) were synthesized by palladium catalysed reaction starting from indole or 7-azaindole using [1,1'-bis(diphenylphosphino)ferrocene]dichloropalladium, as catalyst.

引用

页码：865 / 877

页数：13

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