Cell adhesion integrins as pharmaceutical targets

被引:14
作者
Engleman, VW
Kellogg, MS
Rogers, TE
机构
[1] Searle Research and Development, Monsanto Company, St. Louis, MO 63198
来源
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 31 | 1996年 / 31卷
关键词
D O I
10.1016/S0065-7743(08)60459-5
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:191 / 200
页数:10
相关论文
共 124 条
[11]   RESTRICTED DISTRIBUTION OF INTEGRIN BETA-6 MESSENGER-RNA IN PRIMATE EPITHELIAL TISSUES [J].
BREUSS, JM ;
GILLETT, N ;
LU, L ;
SHEPPARD, D ;
PYTELA, R .
JOURNAL OF HISTOCHEMISTRY & CYTOCHEMISTRY, 1993, 41 (10) :1521-1527
[12]   ASSEMBLY AND FUNCTION OF INTEGRIN RECEPTORS IS DEPENDENT ON OPPOSING ALPHA-CYTOPLASMIC AND BETA-CYTOPLASMIC DOMAINS [J].
BRIESEWITZ, R ;
KERN, A ;
MARCANTONIO, EE .
MOLECULAR BIOLOGY OF THE CELL, 1995, 6 (08) :997-1010
[13]  
BROOKS P, 1995, Patent No. 9525543
[14]   REQUIREMENT OF VASCULAR INTEGRIN ALPHA(V)BETA(3) FOR ANGIOGENESIS [J].
BROOKS, PC ;
CLARK, RAF ;
CHERESH, DA .
SCIENCE, 1994, 264 (5158) :569-571
[15]   ANTIINTEGRIN ALPHA-V-BETA-3 BLOCKS HUMAN BREAST-CANCER GROWTH AND ANGIOGENESIS IN HUMAN SKIN [J].
BROOKS, PC ;
STROMBLAD, S ;
KLEMKE, R ;
VISSCHER, D ;
SARKAR, FH ;
CHERESH, DA .
JOURNAL OF CLINICAL INVESTIGATION, 1995, 96 (04) :1815-1822
[16]   INTEGRIN ALPHA(V)BETA(3) ANTAGONISTS PROMOTE TUMOR-REGRESSION BY INDUCING APOPTOSIS OF ANGIOGENIC BLOOD-VESSELS [J].
BROOKS, PC ;
MONTGOMERY, AMP ;
ROSENFELD, M ;
REISFELD, RA ;
HU, TH ;
KLIER, G ;
CHERESH, DA .
CELL, 1994, 79 (07) :1157-1164
[17]  
BUSK M, 1992, J BIOL CHEM, V267, P5790
[18]  
CARDARELLI PM, 1994, J BIOL CHEM, V269, P18668
[19]   DESIGN AND SYNTHESIS OF NOVEL CYCLIC RGD-CONTAINING PEPTIDES AS HIGHLY POTENT AND SELECTIVE INTEGRIN ALPHA(IIB)BETA(3) ANTAGONISTS [J].
CHENG, S ;
CRAIG, WS ;
MULLEN, D ;
TSCHOPP, JF ;
DIXON, D ;
PIERSCHBACHER, MD .
JOURNAL OF MEDICINAL CHEMISTRY, 1994, 37 (01) :1-8
[20]   INHIBITION OF NEOINTIMAL HYPERPLASIA BY BLOCKING ALPHA(V)BETA(3), INTEGRIN WITH A SMALL PEPTIDE ANTAGONIST GPENGRGDSPCA [J].
CHOI, ET ;
ENGEL, L ;
CALLOW, AD ;
SUN, SP ;
TRACHTENBERG, J ;
SANTORO, S ;
RYAN, US .
JOURNAL OF VASCULAR SURGERY, 1994, 19 (01) :125-134